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A Compendium Of Cyclic Sugar Amino Acids And Their Carbocyclic And Heterocyclic Nitrogen Analogues

Martijn D. P. Risseeuw, M. Overhand, G. Fleet, M. I. Simone
Published 2013 · Chemistry, Medicine

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This compendium focuses on functionalised sugar amino acids (SAAs) and their 3- to 6-membered nitrogen heterocyclic and carbocyclic analogues. The main benefit of using SAAs and their related nitrogen and carbon congeners in the production of peptidomimetics and glycomimetics is that their properties can be readily altered via modification of their ring size, chemical manipulation of their numerous functional groups and fine-tuning of the stereochemical arrangement of their ring substituents. These building blocks provide access to hydrophilic and hydrophobic peptide isosteres whose physical properties allow entry to a region of chemotherapeutic space which is still under-explored by medicinal chemists. These building blocks are also important in providing amino acids whose inherent conformational bias leads to predisposition to secondary structure upon oligomerisation in relatively short sequences. These foldamers, particularly those containing ω-amino acids, provide an additional opportunity to expand access to the control of structures by artificial peptides. The synthesis and biological evaluation of these building blocks in glycomimetics and peptidomimetics systems keep expanding the reach of the glycosciences to the medical sciences, provide a greater outlook onto the wide range of cellular functions of saccharides and their derivatives involved and greater insight into the nature of oligosaccharide and protein folding.
This paper references
10.1016/S0960-894X(02)00467-5
Synthesis and DNA binding properties of saturated distamycin analogues.
C. Woods (2002)
10.1021/JA970855K
Conformational Analysis of Reverse-Turn Constraints by N-Methylation and N-Hydroxylation of Amide Bonds in Peptides and Non-Peptide Mimetics
Y. Takeuchi (1998)
10.1002/CHIN.199924209
Synthesis of an Eight-Carbon Homologue of α-Homomannojirimycin via a Bicyclic Aminolactone.
John P. Shilvock (1999)
10.1021/ja1038819
Tandem 6pi-electrocyclization and cycloaddition of nitrodienes to yield multicyclic nitroso acetals.
Gardner S. Creech (2010)
10.1021/ar700263g
Beta-peptidic peptidomimetics.
D. Seebach (2008)
10.1271/BBB.60.1248
Versatile Synthon for Chirally β-Deuterated L-Amino Acids and Synthesis of (3R)- and (3S)-[3–2H1-l-Serine*
Y. Maeda (1996)
10.1016/J.TETLET.2004.10.064
Synthesis of cyclic oligomers of a modified sugar amino acid utilising dynamic combinatorial chemistry
L. Bornaghi (2004)
10.1039/c1cs15097a
Peptidic foldamers: ramping up diversity.
T. Martinek (2012)
10.1021/JO9702913
Applications of Sugar Nitrones in Synthesis: The Total Synthesis of (+)-Polyoxin J1
A. Dondoni (1997)
10.1002/CBER.19590921008
D‐Galaktosaminuronsäure (2‐Amino‐2‐desoxy‐D‐galakturonsäure) als Baustein des Vi‐Antigens
K. Heyns (1959)
10.1016/J.TETASY.2010.07.010
Esterase-mediated synthesis of optically active GABA analogues containing a stereogenic all-carbon quaternary carbon atom
F. Felluga (2010)
10.1016/S0040-4039(97)01764-4
Peptide-sugar hybrids: Like peptide, like oligosaccharide
Y. Suhara (1997)
10.1002/CHIN.200448099
Metal‐Assisted Synthesis of Enantiopure Spirocyclic β‐Lactams from Azetidine‐2,3‐diones.
B. Alcaide (2004)
10.1111/j.1574-6976.2007.00094.x
Peptidoglycan structure and architecture.
W. Vollmer (2008)
10.1007/s00018-005-5589-y
Sialic acid-specific lectins: occurrence, specificity and function
F. Lehmann (2005)
10.1016/S0968-0896(98)00055-8
Inhibitors of glycogen phosphorylase b: synthesis, biochemical screening, and molecular modeling studies of novel analogues of hydantocidin.
Y. Agasimundin (1998)
10.1021/jo101328c
Unexpected cleavage of 2-azido-2-(hydroxymethyl)oxetanes: conformation determines reaction pathway?
E. Farber (2010)
10.1002/CHIN.200820123
Rapid Access to CF3‐Containing Heterocycles.
A. Dobbs (2008)
10.1002/CHIN.201206119
Catalytic Asymmetric Synthesis of Isoxazoline-N-oxides Through Conjugate Addition—Cyclization under Phase-Transfer Conditions.
T. Kano (2012)
10.1016/J.TETASY.2004.12.024
Efficient synthesis of multifunctional furanoid C-glycoamino acid precursors
Yolanda Vera-Ayoso (2005)
Stereodivergent approach to both syn-and anti-isomers of c-amino-b-hydroxy acids
D Yoo (2011)
Amination of D-mannuronic acid
LG Revelskaya (1973)
10.1016/j.bmc.2008.06.016
Synthesis of both enantiomers of hydroxypipecolic acid derivatives equivalent to 5-azapyranuronic acids and evaluation of their inhibitory activities against glycosidases.
Yuichi Yoshimura (2008)
10.1002/(SICI)1521-3765(20000218)6:4<666::AID-CHEM666>3.0.CO;2-Z
Synthesis and biological evaluation of integrin antagonists containing trans- and cis-2,5-disubstituted THF rings.
F. Osterkamp (2000)
10.1080/07328300600732485
Oxetane δ‐Amino Acids: Chemoenzymatic Synthesis of 2,4‐Anhydro‐5‐N‐(t‐butoxycarbonyl)amino‐D‐lyxonic Acid
Susana Dias Lucas (2006)
10.1271/BBB1961.52.2027
Synthesis of a 2-Amino-2, 5-dideoxy-D-ribofuranoside Analogue
M. Shiozaki (1988)
Novel cyclohexyl-amides
TJ Miles (2011)
10.1021/jo900222g
Stable right- and left-handed peptide helices containing C(alpha)-tetrasubstituted alpha-amino acids.
Andreas A Grauer (2009)
10.1016/S0040-4039(01)01097-8
Diastereospecific formal synthesis of (2R,3S)-2-amino-tetradeca-5,7-dien-3-ol isolated from Xestospongia sp.
N. Langlois (2001)
10.1002/ADSC.200600502
Diversity‐Oriented Preparation of Enantiopure Spirocyclic 2‐Azetidinones from α‐Oxo‐β‐lactams through Barbier‐Type Reactions followed by Metal‐Catalyzed Cyclizations
Benito Alcaide (2007)
10.1021/JO701423W
Tetrahydrofuran Cα-Tetrasubstituted Amino Acids: Two Consecutive β-Turns in a Crystalline Linear Tripeptide
Prantik Maity (2007)
10.1002/EJOC.201001119
Exploitation of Furanoid 5-Azido-3-C-Branched-Chain Sugars Towards Highly Functionalized Nitrogen-Containing Carbohydrate Derivatives
N. Xavier (2011)
3-Amino-2,3-dideoxy-Derythro-furanose derivatives. Tetrahedron
Cheng M-C (1991)
10.1002/CHIN.199830310
Foldamers: A Manifesto
Samuel H. Gellman (1998)
10.1002/CHIN.201223104
Iron-Catalyzed [3 + 2] Annulation of Aminocyclopropanes with Aldehydes: Stereoselective Synthesis of Aminotetrahydrofurans.
F. Benfatti (2012)
10.1016/J.TETASY.2012.03.007
Synthesis of three branched iminosugars [(3R,4R,5S)-3-(hydroxymethyl)piperidine-3,4,5-triol, (3R,4R,5R)-3-(hydroxymethyl)piperidine-3,4,5-triol and (3S,4R,5R)-3-(hydroxymethyl)piperidine-3,4,5-triol] and a branched trihydroxynipecotic acid [(3R,4R,5R)-3,4,5-trihydroxypiperidine-3-carboxylic acid] fr
M. I. Simone (2012)
10.1039/B716835G
Chimeric (α-amino acid + nucleoside-β-amino acid)npeptide oligomers show sequence specific DNA/RNA recognition
K. Gogoi (2008)
10.1002/CHIN.200213113
cis‐ and trans‐3‐Azido‐oxetane‐2‐carboxylate Scaffolds: Hexamers of Oxetane cis‐β‐Amino Acids.
S. F. Barker (2002)
10.1002/HLCA.200390124
Chiral heterospirocyclic 2H-azirin-3-amines as synthons for 3-amino-2,3,4,5-tetrahydrofuran-3-carboxylic acid and their use in peptide synthesis
Simon Stamm (2003)
10.1002/CHIN.200901064
Stereoselective Synthesis and Biological Evaluation of 3,4-Diaminocyclohexanecarboxylic Acid Derivatives as Factor Xa Inhibitors.
T. Nagata (2009)
10.1002/ANGE.19780901030
Funktionelle D‐ und L‐Ribose‐Derivate über eine Racematspaltung mit Rückführung
R. Schmidt (1978)
10.1016/S0040-4020(01)89766-0
Asymmetric synthesis of malic acid-type synthons VIA chiral norephedrine-derived oxazolidines
A. Bernardi (1990)
10.1248/CPB.14.537
Studies on Optically Active Amino Acids. VIII. Studies on α-Alkyl-α-amino Acids. III. Determination of Absolute Configuration of Optically Active Isovaline.
K. Achiwa (1966)
10.1021/JO060296C
Formal total synthesis of the potent renin inhibitor aliskiren: application of a SmI2-promoted acyl-like radical coupling.
Karl B. Lindsay (2006)
10.1039/b714350h
Peptides derived from nucleoside beta-amino acids form an unusual 8-helix.
R. Threlfall (2008)
10.1016/J.TETASY.2003.12.034
Synthesis of enantiopure 1,4-ethyl- and 1,4-ethylene-bridged cispentacin by lipase-catalyzed enantioselective ring opening of β-lactams
E. Forró (2004)
10.1002/CHIN.201317235
Spirocyclic Nucleosides in Medicinal Chemistry: An Overview
R. Soengas (2013)
10.1021/JM960155A
Synthesis of a series of aryl kainic acid analogs and evaluation in cells stably expressing the kainate receptor humGluR6.
B. Cantrell (1996)
10.1016/J.TETASY.2004.07.032
Oxetane cis- and trans-β-amino-acid scaffolds from l-rhamnose by efficient SN2 reactions in oxetane rings; pseudoenantiomeric analogues of the antibiotic oxetin
S. Johnson (2004)
10.1016/J.BMCL.2006.11.020
Design and synthesis of a novel class of furan-based molecules as potential 20S proteasome inhibitors.
Yiqiu Fu (2007)
10.3390/11070564
Novel furanoid alpha-substitued alpha-amino acid as a potent turn mimic in peptide synthesis.
M. Martinková (2006)
10.1021/JO7018762
Synthesis of epi-oxetin via a serine-derived 2-methyleneoxetane.
M. L. Blauvelt (2008)
10.1039/P19910001637
Structural elucidation and solution conformation of the novel herbicide hydantocidin
H. Haruyama (1991)
10.1016/S0040-4039(99)00111-2
An octameric carbopeptoid; secondary structure in octameric and tetrameric 5-aminomethyl-tetrahydrofuran-2-carboxylates
T. Claridge (1999)
10.1016/0040-4039(80)80077-3
Total Synthesis of 2,4-methanaproline
M. Pirrung (1980)
10.1016/0040-4039(91)80016-Y
Stereoselective epoxidation of chiral electron-poor γ-aminoolefins
M. T. Reetz (1991)
10.1039/B105111N
β-Aminophosphonic compounds derived from methyl 1-dimethoxyphosphoryl-2-succinimidocyclohex-3-ene-1-carboxylates
Nathalie Defacqz (2001)
10.1016/S0040-4039(02)00689-5
Novel conformationally restricted glycoamino acids from glyco-α-aminonitriles as potent turn mimics in peptide synthesis
A. N. V. Nhien (2002)
10.1002/CHIN.200022177
Synthesis of Nojirimycinyl C‐(L)‐Serine.
T. Fuchß (2000)
10.1016/J.TET.2011.12.052
Sulfanyl-methylene-5(4H)-oxazolones and β-sulfanyl-α-nitroacrylates as appealing dienophiles for the synthesis of conformationally constrained cysteine analogues
Alessandro Ruffoni (2012)
10.1002/CHIN.199548221
A Versatile Approach to Acromelic Acid Analogues.
J. Baldwin (1995)
10.1016/S0040-4039(03)01416-3
Synthesis of all diastereomeric methyl 2,5-anhydro-3-deoxy-hexonates: precursors to C-2-deoxynucleosides and THF-templated γ- and δ-amino acids
M. Watterson (2003)
10.1021/JA068455X
Total synthesis of plusbacin A3: a depsipeptide antibiotic active against vancomycin-resistant bacteria.
Aaron M. Wohlrab (2007)
10.1016/0040-4039(96)00094-9
Synthesis of a new carbohydrate mimetics: “carbopeptoid” containing a C-1 carboxylate and C-2 amino group
Y. Suhara (1996)
10.1002/CHIN.200306186
Synthesis of Nojirimycin C‐Glycosides.
L. Cipolla (2003)
10.1002/CHIN.199811290
β‐Peptides: A Surprise at Every Turn
D. Seebach (1998)
10.1002/CHIN.199706197
Synthesis and Conformational Analysis of Linear and Cyclic Peptides Containing Sugar Amino Acids.
E. V. Roedern (1997)
10.1055/S-2006-941573
You Are Sitting on a Gold Mine
C. Toniolo (2006)
10.1016/0223-5234(89)90086-X
Synthèse des deux énantiomères de l'analogue carbocyclique du nicotinamide ribose et évaluation de leurs propriétés biologiques
M. Ikbal (1989)
10.1080/07328319608002388
A Novel Type of Spironucleosides: 2′,5′-O-bis-TBDMS Uridine-3′-spiro-3′-isoxazolidin-5′-one and Its Thymidine Congener +
J. Tronchet (1996)
10.1016/J.BMCL.2005.08.109
Synthesis and evaluation of novel 8,6-fused bicyclic peptidomimetic compounds as interleukin-1β converting enzyme inhibitors
S. V. O'neil (2005)
10.1021/JO035199N
Modification of 1-substituents in the 2-azabicyclo[2.1.1]hexane ring system; approaches to potential nicotinic acetylcholine receptor ligands from 2,4-methanoproline derivatives.
J. Malpass (2003)
10.1016/0008-6215(91)84042-D
Thermal and photochemical degradation of sodium N-acetylneuraminate
N. Sugiyama (1991)
10.1039/B517883E
Syntheses and bio-activities of the L-enantiomers of two potent transition state analogue inhibitors of purine nucleoside phosphorylases.
K. Clinch (2006)
10.1016/J.TETLET.2006.09.005
A β-lactam-azasugar hybrid as a competitive potent galactosidase inhibitor
G. Pandey (2006)
10.1002/CHIN.200135209
Isolation, Structure Determination, and Synthesis of Neodysiherbaine A, a New Excitatory Amino Acid from a Marine Sponge.
R. Sakai (2001)
10.1021/cc700171p
"Diversity oriented synthesis" of functionalized chiral tetrahydropyridines: potential GABA receptor agonists and azasugars from natural amino acids via a sequential Baylis-Hillman reaction and RCM protocol.
P. R. Krishna (2008)
10.1016/j.bmc.2009.10.023
Design, synthesis, and SAR of cis-1,2-diaminocyclohexane derivatives as potent factor Xa inhibitors. Part I: exploration of 5-6 fused rings as alternative S1 moieties.
K. Yoshikawa (2009)
10.1021/JA963036T
Influenza neuraminidase inhibitors possessing a novel hydrophobic interaction in the enzyme active site: design, synthesis, and structural analysis of carbocyclic sialic acid analogues with potent anti-influenza activity.
C. U. Kim (1997)
10.1039/B211642A
Diastereoselective titanium-mediated construction of cis-2,3-ring annelated 1-(2'-chloroethyl)cyclopropanols.
F. Lecornué (2003)
10.1039/B709627E
A highly stereocontrolled total synthesis of dysiherbaine.
K. Takahashi (2007)
10.1111/j.1574-6976.2008.00114.x
Structure and genetics of Shigella O antigens.
B. Liu (2008)
10.1016/S0040-4039(00)99490-5
Design and synthesis of substrate analogs for the inhibition of dehydroquinate synthase
Nicholas Nikolaides (1989)
A short synthesis of 2,3diacetamido-2,3-dideoxy-D-mannuronic acid-derivatives
AG Hedenetz (2000)
10.1016/J.TETASY.2008.12.017
Stereocontrolled transformation of nitrohexofuranoses into cyclopentylamines via 2-oxabicyclo[2.2.1]heptanes. III: synthesis of enantiopure methyl (1S,2S,3R,4S,5R)-2-amino-3,4,5-trihydroxycyclopentanecarboxylate
F. Fernandez (2008)
10.1002/1099-0690(200104)2001:8<1541::AID-EJOC1541>3.0.CO;2-7
Synthesis and structural analysis of a beta-hairpin peptide containing a sugar amino acid
Begoña Aguilera (2001)
10.1039/A904064A
Synthesis of homorhamnojirimycins and related trihydroxypipecolic acid derivatives via divergent bicyclic amino lactone intermediates: Inhibition of naringinase (L-rhamnosidase) and dTDP-rhamnose biosynthesis
John P. Shilvock (1999)
10.1002/EJOC.200700333
Synthetic Routes to Three Novel Scaffolds for Potential Glycosidase Inhibitors
M. Rommel (2007)
10.1351/goldbook.s05990
Stereoselective Synthesis of (
An (2001)
10.1021/OL0514707
Selective Michael-aldol reaction by use of sterically hindered aluminum aryloxides as Lewis acids: an easy approach to cyclobutane amino acids.
A. Avenoza (2005)
10.1055/S-2004-820031
Iodine-mediated Ring Closing Alkene Iodoamination with N-Debenzylation for the Asymmetric Synthesis of Polyhydroxylated Pyrrolidines
S. Davies (2004)
10.1016/0040-4039(95)00198-L
Spirohydantoins of glucofuranose: Analogues of hydantocidin
Tilmann W. Brandstetter (1995)
10.1016/S0957-4166(00)00284-6
Carbocyclic α-amino acids: asymmetric Strecker synthesis of a series of 2-alkylated 1-aminocyclopentanecarboxylic acids
Judith Wede (2000)
10.1021/JO9909397
STEREOSELECTIVE MANNICH-TYPE REACTION OF AN ACYCLIC KETIMINE WITH A SUBSTITUTED CHLOROTITANIUM ENOLATE : EFFICIENT APPROACH TO D-ERYTHRO-ALPHA -TRIFLU OROMETHYL-BETA -HYDROXYASPARTIC UNITS
P. Bravo (1999)
10.1246/BCSJ.62.3950
Synthesis of 2-Amino-2-deoxy-α-D-altrofuranoside Derivatives from 2,3-O-Isopropylidene-D-glyceraldehyde via Bicyclic β-Lactam Intermediates
M. Shiozaki (1989)
10.1002/CHIN.197717346
SYNTHESIS OF 9‐AZAPROSTAGLANDIN ANALOGS
G. P. Rozing (1976)
10.1002/CHIN.200119123
Selective Fowler Reductions: Asymmetric Total Syntheses of Isofagomine and Other 1-Azasugars from Methyl Nicotinate.
G. Zhao (2001)
10.1002/CHIN.200025248
Synthesis of (‐)‐Dysiherbaine.
B. B. Snider (2000)
10.1002/(SICI)1522-2675(19991006)82:10<1559::AID-HLCA1559>3.0.CO;2-A
Synthesis, Crystal Structures, and Modelling ofβ-Oligopeptides Consisting of 1-(Aminomethyl)cyclopropanecarboxylic Acid: Ribbon-Type Arrangement of Eight-Membered H-Bonded Rings
S. Abele (1999)
10.1002/PSC.658
Conformational studies of oligomeric oxetane‐based dipeptide isosteres derived from L‐rhamnose or D‐xylose
Stephen W. Johnson (2005)
10.1016/j.bmc.2010.06.091
Design, synthesis, and biological evaluation of conformationally constrained glycerol 3-phosphate acyltransferase inhibitors.
Edward A Wydysh (2010)
10.1002/anie.201101301
Characteristic structural parameters for the γ-peptide 14-helix: importance of subunit preorganization.
L. Guo (2011)
10.1002/CHIN.200212235
A Bioisosteric Oligosaccharide Mimetic Based on Isofagomine‐Type Monomers.
Xifu Liang (2002)
10.1016/S0040-4039(00)61520-4
Highly substituted cis-β-cyclopentane amino acids : an approach to the synthesis of trehazolin analogues
R. Elliott (1993)
10.1002/EJOC.200300554
3-Aminobicyclo[1.1.1]pentane-1-carboxylic Acid Derivatives: Synthesis and Incorporation into Peptides
M. Pätzel (2004)
10.1021/JM00378A023
Peptide sweeteners. 6. Structural studies on the C-terminal amino acid of L-aspartyl dipeptide sweeteners.
J. Tsang (1984)
10.1021/JO0495034
concise synthesis of 4-acylamino analogues of 2-aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acids (LY354740) from an acylnitroso Diels-Alder cycloadduct.
W. Lee (2004)
10.1016/S0040-4039(00)78525-X
Tri- and tetra-peptides incorporating an α-amino acid at the anomeric position of mannofuranose
J. Estévez (1994)
10.1016/S0040-4020(01)00530-0
Facile synthesis and highly efficient resolution of a constrained cyclopropane analogue of phenylalanine
A. Jimenez (2001)
10.1016/j.bmc.2011.12.046
Quinolone derivatives containing strained spirocycle as orally active glycogen synthase kinase 3β (GSK-3β) inhibitors for type 2 diabetics.
S. Seto (2012)
10.1016/J.TET.2007.05.066
Adamantane-retropeptides, new building blocks for molecular channels
N. Basarić (2007)
10.3762/bjoc.7.94
Homoallylic amines by reductive inter- and intramolecular coupling of allenes and nitriles
P. Wipf (2011)
10.1016/J.TETASY.2004.11.034
Stereocontrolled transformation of nitrohexofuranoses into cyclopentylamines via 2-oxabicyclo[2.2.1]heptanes. Part 2: Synthesis of (1S,2R,3S,4S,5R)-3,4,5-trihydroxy-2-aminocyclopentanecarboxylic acid
R. Soengas (2005)
10.1016/J.TETASY.2009.09.001
Efficient synthesis of 3,4- and 4,5-dihydroxy-2-amino-cyclohexanecarboxylic acid enantiomers
Gabriella Benedek (2009)
10.1016/S0040-4039(00)78528-5
Aldol equilibrations of unprotected trihydroxybicyclic lactones: Enantiomeric tetrahydroxy-α-aminocyclopentane carboxylic acids from epimeric bicyclic lactones
Andrew Hui (1994)
10.1002/EJOC.200600068
Tetrahydropyran‐Amino Acids: Novel Building Blocks for Gramicidin‐Hybrid Ion Channels
S. Schröder (2006)
10.1002/ADSC.200900879
Asymmetric Synthesis of 2,3,4-Trisubstituted Functionalised Tetrahydrofurans via an Organocatalytic Michael Addition as Key Step
D. Enders (2010)
10.1016/J.TET.2004.07.032
Conformational studies of 3,4-dideoxy furanoid sugar amino acid containing analogs of the receptor binding inhibitor of vasoactive intestinal peptide
T. Chakraborty (2004)
Enantionselective synthesis of Loracarbef from sodium erythrobate
JW Frazier (1992)
10.1081/CAR-120016491
PYRANOSYL SUGAR AMINO ACID CONJUGATES: THEIR BIOLOGICAL ORIGINS, SYNTHETIC PREPARATIONS, AND STRUCTURAL CHARACTERIZATION
J. Gervay-Hague (2002)
10.1021/ol200567p
Large-scale asymmetric synthesis of the bioprotective agent JP4-039 and analogs.
Marie-Céline Frantz (2011)
10.1002/ANIE.200460420
Chiral Centers in the Side Chains of α‐Amino Acids Control the Helical Screw Sense of Peptides
M. Tanaka (2004)
2008a) a, b-Cyclic-b-benzamido hydroxamic acids: novel templates for the design, synthesis, and evaluation of selective inhibitors of TNF-a converting enzyme (TACE)
Gr Ott
10.1002/CHIN.199916200
Preparation and Structure of β‐Peptides Consisting of Geminally Disubstituted β2,2‐ and β3,3‐Amino Acids: A Turn Motif for β‐Peptides.
D. Seebach (1999)
10.1002/CBER.191304603125
Über Tetraamino‐adipinsäure und β,β′‐Diamino‐α,α′‐dioxyadipinsäure
W. Traube (1913)
10.1002/CHIN.199024318
Synthesis of Homochiral β-Hydroxy-α-amino Acids ((2S,3R,4R)-3,4-Dihydroxyproline and (2S,3R,4R)-3,4-Dihydroxypipecolic Acid) and of 1,4-Dideoxy-1,4-imino-D-arabinitol (DAB1) and Fagomine (1,5-Imino-1,2,5-trideoxy-D-arabino-hexitol).
G. W. J. Fleet (1990)
10.1002/CHIN.200103116
Claisen Rearrangement of Allylic Alcohols Prepared Through N‐Boc‐2‐acyloxazolidine Methodology. Application to the Synthesis of Trisubstituted Cyclopropanes.
C. Agami (2001)
10.1055/S-2003-38058
Indium-mediated allylation reaction in aqueous media: Synthetic studies towards the total synthesis of dysiherbaine
Jing-Mei Huang (2003)
10.1248/CPB.28.2337
Medicinal chemical studies on antiplasmin drugs. VIII. 4-Aminomethylcyclohexanecarboxylic acid derivatives having a carboxyl or carboxymethyl group at C2.
S. Isoda (1980)
10.1016/J.TETASY.2006.06.032
Creation of quarternary stereocentres via [3,3]-sigmatropic rearrangement of allylic thiocyanates. A synthetic approach to (+)-myriocin
J. Gonda (2006)
10.1016/S0040-4039(00)60117-X
Novel L-Phe-Gly mimetics
Li Yi-Lin (1992)
Discovery of potent and selective inhibitors of 11beta-HSD1 for the treatment of metabolic syndrome.
Steven Richards (2006)
10.1021/jo801123q
Synthesis, conformational analysis and biological studies of cyclic cationic antimicrobial peptides containing sugar amino acids.
T. Chakraborty (2008)
10.1002/CHIN.200616248
Carbohydrates in Peptide and Protein Design
K. J. Jensen (2006)
10.1016/J.TET.2004.01.030
Anomeric spiroannelated 1,4-diazepine 2,5-diones from furano exo-glycals: towards a new class of spironucleosides
C. Taillefumier (2004)
10.1016/J.TET.2007.12.032
A general and efficient stereoselective synthesis of γ-azido-tetrahydrofuran carboxylic acids from glycals
P. V. Reddy (2008)
10.1039/B002995P
Tetrahydrofuran amino acids—versatile building blocks for unnatural biopolymers: lack of secondary structure in oligomeric carbopeptoids derived from a D-galacto-5-(aminomethyl) tetrahydrofuran-2-carboxylic acid
D. Brittain (2000)
10.1039/A807313I
β-Hydroxypiperidinecarboxylates: additions to the chiral pool from bakers’ yeast reductions of β-ketopiperidinecarboxylates
D. Knight (1998)
10.1055/S-2000-6251
Synthesis of Nojirimycinyl C-(l)-Serine
T. Fuchs (2000)
10.1055/S-2005-922768
Synthesis of spirocyclic glucose-proline hybrids (GlcProHs)
Kaidong Zhang (2005)
10.1016/0957-4166(96)00014-6
Mimics of l-rhamnose: Analogues of rhamnopyranose containing a constituent α-amino acid at the anomeric position. A rhamnopyranose analogue of hydantocidin
J. Estévez (1996)
10.1002/CHIN.199628107
Synthesis of (1′S,3′R)‐3‐(3′‐Amino‐2′,2′‐dimethylcyclobutyl)propan‐1‐ ol from (‐)‐β‐Pinene.
J. Blanco (1996)
10.1016/0008-6215(94)00313-5
Synthesis of methyl (d-glycopyranosyl azide) uronates
Z. Gyoergydeak (1995)
10.1080/00397911.2010.491595
Expedient Synthesis of cis- and trans-3-Aminocyclobutanecarboxylic Acids
D. Radchenko (2011)
10.1021/jo1024915
Silver-catalyzed 1,3-dipolar cycloaddition of azomethine ylides with β-boryl acrylates.
A. López-Pérez (2011)
10.1021/JO00085A036
Reductive cyclization of ketones tethered to activated olefins mediated by magnesium in methanol
G. Lee (1994)
A compendium of cyclic sugar amino acids 685
Synthesis of a new carbohydrate mimetics "carbopeptoid"
Suhara Suhara (1996)
10.1016/S0040-4039(01)81580-X
Enantiospecific synthesis of (s)-4-amino-4,5-dihydro-2-furancarboxylic acid, a new suicide inhibitor of gaba-transaminase.
J. P. Burkhart (1984)
10.1016/S0957-4166(99)00045-2
Carbocyclic α-amino acids: asymmetric synthesis of all four 1-amino-2-hydroxycyclohexanecarboxylic acids
K. P. Fondekar (1999)
10.1002/CHIN.200102108
Tetrahydrofuran as a Scaffold for Peptidomimetics. Application to the Design and Synthesis of Conformationally Constrained Metalloproteinase Inhibitors.
S. Hanessian (2001)
10.1021/JA01544A038
The Alkaloids of Tabernanthe Iboga. VII.1 Derivatives of Isoquinuclidine
L. Werner (1958)
1975a) Polysaccharidanaloga I
Fuchs E-F (1975)
10.1081/SCC-120023992
A Practical Process for the Preparation of Azetidine-3-carboxylic Acid
R. A. Miller (2003)
10.1002/CHIN.198731328
Synthesis of Azacyclic 2-Deoxy-KDO (I).
D. W. Norbeck (1987)
10.1016/0040-4020(96)00949-0
Synthesis of chiral nonracemic homo-1-deoxyazasugars with D-talo-and L-allo-configuration via tandem Wittig [2+3] cycloaddition reaction
C. Herdeis (1996)
10.1016/J.TETASY.2010.06.026
Stereochemistry of terpene derivatives. Part 7: Novel rigidified amino acids from (+)-3-carene designed as chiral GABA analogues☆
K. Gajcy (2010)
10.1021/CC034054R
Tetrahydrofuran-based amino acids as library scaffolds.
A. A. Edwards (2004)
10.1021/OL027229Z
Toward amide-linked RNA mimics: total synthesis of 3'-C branched uridine azido acid via an ene-iodolactonization approach.
E. Rozners (2003)
10.1021/JO951983Z
Synthesis of Optically Pure 3,4-Disubstituted l-Glutamates from a Novel 2,3-Aziridino-γ-lactone 4-Carboxylate Derivative
Philippe Dauban (1996)
10.1002/CHIN.200136185
Novel and Efficient Transformation of α-Amino Nitrile to α-Imino and α-Amide Nitriles in Asymmetric Strecker Synthesis.
K. Namba (2001)
10.1021/ol2028459
Expanding the azaspiro[3.3]heptane family: synthesis of novel highly functionalized building blocks.
Johannes A. Burkhard (2012)
10.1039/JR9310001382
CLXXXVI.—Some reactions of ortho-derivatives of aldehydes and ketones
W. Cocker (1931)
10.1107/S0108270194010656
(2S,3R,4S)-4-(1,1-Dimethylethoxycarbonylamino)-2,3-epoxy-5-phenylpentanoic acid ethyl ester
H. Weber (1995)
10.1002/CHIN.199450220
Asymmetric Synthesis of the Natural Diastereoisomer of trans-α-( 2-Carboxymethylcyclopropyl)glycine Isolated from Blighia unijugata.
C. Alcaraz (1994)
10.1016/S0040-4020(00)01023-1
New synthesis of 7-azabicyclo[2.2.1]heptane-1-carboxylic acid
A. Avenoza (2001)
10.1002/asia.200900033
Metal-catalyzed derivatization of C(alpha)-tetrasubstituted amino acids and their use in the synthesis of cyclic peptides.
A. Grauer (2009)
10.1021/JO034940O
Synthesis of cyclic and acyclic beta-amino acids via chelation-controlled 1,3-dipolar cycloaddition.
R. Hanselmann (2003)
derived-b-amino acid sequences
A Ghorai (2011)
10.1021/JO0110698
Design, synthesis, and evaluation of matrix metalloprotease inhibitors bearing cyclopropane-derived peptidomimetics as P1' and P2' replacements.
A. Reichelt (2002)
10.1016/S0960-894X(02)00520-6
Synthesis and preliminary evaluation of trans-3,4-conformationally-restricted glutamate and pyroglutamate analogues as novel EAAT2 inhibitors.
T. Denton (2002)
10.1016/0040-4020(80)80071-8
Heteroatom directed photoarylation synthesis of functionalized indolines
A. G. Schultz (1980)
10.1074/jbc.M112.369561
Lipodepsipeptide Empedopeptin Inhibits Cell Wall Biosynthesis through Ca2+-dependent Complex Formation with Peptidoglycan Precursors*
Anna Müller (2012)
10.1002/CHIN.200246190
Design and Synthesis of a Novel Class of Sugar‐Peptide Hybrids: C‐Linked Glyco β‐Amino Acids Through a Stereoselective “Acetate” Mannich Reaction as the Key Strategic Element.
C. Palomo (2002)
10.1016/J.TETASY.2009.12.018
Studies on the stereocontrolled transformation of nitrohexofuranoses into 2-oxabicyclo[2.2.1]heptanes. V: Synthesis of enantiopure methyl (1R,2R,4S)-2-amino-4-hydroxycyclopentanecarboxylate
A. Estévez (2010)
10.1039/B002997L
Tetrahydrofuran amino acids: β- and γ-azidotetrahydrofurancarboxylic acid monomers derived from D-glucoheptonolactone as building blocks for β- and γ-oligopeptides
N. Hungerford (2000)
10.1002/CHIN.199008367
Muramylpeptides and Lipopeptides: Studies Towards Immunostimulants
G. Baschang (1990)
10.1039/B719451J
Simple and quantitative mechanochemical preparation of the first zinc and copper complexes of the neuroleptic drug gabapentin
D. Braga (2008)
10.1016/J.TETLET.2006.11.146
First total synthesis of penmacric acid and its stereoisomer
M. Ueda (2007)
10.1016/0040-4020(96)00594-7
α-Azidoesters as divergent intermediates for combinatorial generation of glucofuranose libraries of novel N-linked glycopeptides
Tilmann W. Brandstetter (1996)
10.1021/BI00136A012
Helical epitope of the group B meningococcal alpha(2-8)-linked sialic acid polysaccharide.
J. Brisson (1992)
10.1016/S0040-4039(00)78527-3
Polyhydroxylated cyclohexane and cyclopentane α-amino acids from cyclisations of an azidolactone
A. Fairbanks (1994)
10.1002/CHIN.200224131
Claisen Rearrangements of Allylic and Propargylic Alcohols Prepared by an N-Boc-2-acyloxazolidine Methodology — Application to the Synthesis of Original Chiral Building Blocks.
C. Agami (2010)
10.1021/JO00103A057
A GENERAL SYNTHETIC ROUTE TO ANOMERIC ALPHA -AZIDO AND ALPHA -AMINO ACIDS AND FORMAL SYNTHESIS OF ()-HIDANTOCIDIN
A. Dondoni (1994)
10.1016/J.TET.2006.08.006
Efficient synthesis of a new pipecolic acid analogue with a bicyclic structure
D. Casabona (2006)
10.1016/S0040-4020(01)85738-0
Synthesis of highly functionalized homochiral azetidines and azetidine-2-carboxylic esters
A. Duréault (1993)
10.1021/JO00109A004
A New Asymmetric Synthesis of .alpha.-Methylcysteines via Chiral Aziridines
H. Shao (1995)
10.1016/S0040-4039(00)82143-7
Synthesis of both epimeric 2-deoxy-N-acetylneuraminic acids and their behaviour towards CMP-sialate synthetase: a comparison with 2-β-methylketoside of N-acetylneuraminic acid
W. Schmid (1988)
10.1021/ol3008815
New preorganized γ-amino acids as foldamer building blocks.
Li Guo (2012)
10.1002/CHIN.199051359
Synthesis of Optically Pure Analogues of D-Arginine Methyl Ester with Antiarrhythmic Activity.
A. Banfi (1990)
10.1002/EJOC.200210682
Synthesis of Novel Sugar Amino Acids by Curtius Rearrangement
R. V. Well (2003)
Synthesis of nucleosides and related-compounds. 36. Explanation for stereoselectivity of the cis-dihydroxylation of cis-3,5-disubstituted cyclopentenes
N Katagiri (1994)
10.1016/J.TETASY.2007.09.028
Regio- and stereoselective synthesis of the enantiomers of monoterpene-based β-amino acid derivatives
Zsolt Szakonyi (2007)
10.1002/chem.201001108
High-yielding synthesis of the anti-influenza neuraminidase inhibitor (-)-oseltamivir by two "one-pot" sequences.
H. Ishikawa (2010)
10.1039/c1ob06095c
Stereoselective preparation of β,γ-methano-GABA derivatives.
D. Aitken (2011)
A novel type of spironucleosides: 2 0 ,5 0 -O-bis-TBDMS uridine-3 0 - spiro-3 0 -isoxazolidin-5 0 -one and its thymidine congener
Jmj Tronchet (2006)
10.1016/S0022-1139(00)80382-6
Darstellung von 1-amino-3-trifluormethyl-adamantan
R. Feldhoff (1990)
10.1104/pp.110.3.753
Adenylosuccinate Synthetase: Site of Action of Hydantocidin, a Microbial Phytotoxin
D. Siehl (1996)
10.1002/EJOC.200500297
Synthesis of 3-and 4-hydroxy-2-aminocyclohexanecarboxylic acids by iodocyclization
Zsolt Szakonyi (2005)
10.1002/chin.198623334
A Chiral Nitronate Dianion from D-Glyceraldehyde. Enantiospecific Syntheses of 2,3-Dideoxy-3-nitro Furanosides and Pyranosides.
T. M. Williams (1986)
10.1002/CHIN.200044231
Stereospecific Synthesis of Two Novel Cytotoxic Pyrazole C‐Nucleosides from D‐Glucose.
M. Popsavin (2000)
10.1021/JO00310A010
THE TOTAL SYNTHESIS OF NIKKOMYCIN B
A. Barrett (1990)
10.1002/cmdc.201200541
3‐Hydroxyazetidine Carboxylic Acids: Non‐Proteinogenic Amino Acids for Medicinal Chemists
Andreas F. G. Glawar (2013)
10.1016/S0957-4166(02)00473-1
Facile synthesis of fused furanosyl β-amino acids from protected sugar lactones: incorporation into a peptide chain
C. Taillefumier (2002)
10.1039/A907655G
Anionically induced decomposition of ethyl 2-(2,2-dimethylethylperoxymethyl)propenoate by amines: an easy access to amino epoxyesters and amino ester peroxides
C. Cramay (1999)
10.1016/S0008-6215(00)83144-4
The synthesis of 5-amino-2,6-anhydro-5-deoxy-D-glycero-D-gulo-Heptonic acid and its polycondensation to oligomers
E. Fuchs (1976)
10.1016/j.ejmech.2011.04.011
Second-generation sulfonamide inhibitors of D-glutamic acid-adding enzyme: activity optimisation with conformationally rigid analogues of D-glutamic acid.
Izidor Sosič (2011)
10.1002/CHIN.200446217
Enantioselective Synthesis of (-)-Galantinic Acid.
S. Pandey (2004)
10.1016/J.TET.2006.03.038
Synthesis and DNA binding studies of bis-intercalators with a novel spiro-cyclic linker
Yongjun Chu (2006)
Advances in Amino Acid Mimetics and Peptidomimetics
A. Abell (1997)
10.1002/CHIN.199605307
Synthesis of Complex Nucleoside Antibiotics
S. Knapp (1996)
10.1248/CPB.28.1408
Medicinal Chemical Studies on Antiplasmin Drugs. VI. Aza Analogs of 4-Aminomethylbenzoic Acid
S. Isoda (1980)
a, c-Cyclic peptide ensembles with a hydroxylated cavity
C Reiriz (2009)
10.1055/S-1993-22344
The Wittig Reaction of Moncyclic β-Lactams
J. Baldwin (1993)
10.1021/JM051026+
Tumor-cell-targeted methionine-enkephalin analogues containing unnatural amino acids: design, synthesis, and in vitro antitumor activity.
Š. Horvat (2006)
10.1039/B108310D
A novel stereoselective synthesis of N-heterocycles by intramolecular hydrovinylation
U. Bothe (2001)
10.1107/S1600536805001467
(3R,4R,5S)-5-(Acetamido­methyl)-N-benzyl-3,4-dihydroxy­tetrahydro­furan-3-carboxamide
F. Punzo (2005)
10.1021/JM0255724
3'-Aminoadenosine-5'-uronamides: discovery of the first highly selective agonist at the human adenosine A3 receptor.
M. Deninno (2003)
10.1016/S0040-4039(99)00389-5
2′-deoxyribo-PNAs: A structurally novel class of polyamide nucleic acids with good RNA and DNA binding affinity
P. Matt (1999)
10.1021/jo101763t
Synthesis and structural studies of homooligomers of geminally disubstituted β(2,2)-amino acids with carbohydrate side chain.
G. V. M. Sharma (2011)
10.1002/CHIN.199628249
Nucleophilic Opening of Epoxide by Guanidine. A Route to Potential Substrates or Inhibitors of NO Synthases.
C. Gravier-Pelletier (1996)
10.1055/S-1989-34699
Stereoselective Cycloadditions of Chiral Acyl-Nitroso Compounds
A. Miller (1989)
New potent, orally active neuraminidase inhibitors as anti-influenza agents: in vitro and in vivo activity of GS4071 and analogs
CU Kim (1996)
10.1002/CHIN.200347078
Synthesis of Polyhydroxylated Aminocyclopentanes.
Markus Kummeter (2003)
10.1021/JO0621874
Rapid synthesis of cyclodepsipeptides containing a sugar amino acid or a sugar amino alcohol by a sequence of a multicomponent reaction and acid-mediated macrocyclization.
Carine Bughin (2007)
A compendium of cyclic sugar amino acids 689
10.1016/J.TETLET.2003.12.032
Synthesis of pyranoid δ-sugar amino acids and their oligomers from per-benzylated β-C-vinyl glucoside
François Durrat (2004)
Synthesis of C
Tomoya Aoba (2013)
10.1021/JO052506B
5-Carboxy-2-azabicyclo[2.1.1]hexanes as precursors of 5-halo, amino, phenyl, and 2-methoxycarbonylethyl methanopyrrolidines.
G. Krow (2006)
10.1016/J.TETASY.2003.11.022
Stereoselective synthesis of novel tetrahydroxypyrrolizidines
Ana T Carmona (2004)
10.1016/S0040-4039(00)72710-9
Preparation of heterocyclic amino acids via intramolecular mukaiyama aldol condensation: Synthesis of a novel cycloleucine analogue
D. M. Walker (1989)
10.1016/j.ejmech.2011.02.061
Design and synthesis of protein-protein interaction mimics as Plasmodium falciparum cysteine protease, falcipain-2 inhibitors.
L. Rizzi (2011)
10.1071/CH03214
An Alternative Synthesis of Some Carbohydrate α-Amino Acids
Grant S. Forman (2004)
10.1021/OL0166698
Sugar amino acid containing somatostatin analogues that induce apoptosis in both drug-sensitive and multidrug-resistant tumor cells.
S. Gruner (2001)
10.1002/CHIN.200110257
Novel Synthesis of (+)-4-Acetoxy-3-hydroxyethyl-2-azetidinone from Carbohydrate. A Formal Total Synthesis of (+)-Thienamycin.
K. Tatsuta (2001)
10.1021/ol2022356
Simultaneous parallel and antiparallel self-assembly in a triazole/amide macrocycle conformationally homologous to D-,L-α-amino acid based cyclic peptides: NMR and molecular modeling study.
A. Ghorai (2011)
10.1016/J.TETLET.2005.06.029
Branched tetrahydrofuran α,α-disubstituted-δ-sugar amino acid scaffolds from branched sugar lactones: a new family of foldamers?
M. I. Simone (2005)
10.1016/J.TETLET.2004.04.013
Stereoselective synthesis of novel conformationally restricted β- and γ-amino acids
Frieder Gnad (2004)
10.1021/JM0110486
(2S,1'S,2'S,3'R)-2-(2'-carboxy-3'-methylcyclopropyl) glycine is a potent and selective metabotropic group 2 receptor agonist with anxiolytic properties.
I. Collado (2002)
10.1007/s00726-010-0690-4
An efficient route towards a new branched tetrahydrofurane δ-sugar amino acid from a pyrolysis product of cellulose
A. Defant (2010)
10.1021/JA00229A048
Synthesis of (-)-oxetanocin
D. Norbeck (1988)
10.1007/s00044-010-9498-8
Synthesis and biological activities of Schiff bases of gabapentin with different aldehydes and ketones: a structure–activity relationship study
L. Mallesha (2010)
10.1002/CHEM.19970030614
Synthesis and biological evaluation of a backbone-modified phytoalexin elicitor
C. M. Timmers (1997)
Deoxyiminoalditols from aldonolactones: 1. Preparation of 1,4-dideoxy-1,4-iminohexitols with D-allo and L-allo and D-talo and L-talo configuration—potential glycosidase inhibitors
I Lundt (1993)
10.1016/S0040-4039(00)78526-1
Spirocyclic peptides at the anomeric position of mannofuranose
J. C. Estévez (1994)
10.1016/j.bmcl.2010.09.028
Design, synthesis, and structure-activity relationship studies of N-arylsulfonyl morpholines as γ-secretase inhibitors.
H. Li (2010)
10.1016/0040-4039(91)80836-U
Approach to oxetane and furan nucleosides with an anomeric carbon substituent : nucleophilic substitution at highly hindered α-bromo-oxetane- and -tetrahydrofuran-carboxylates
S. Choi (1991)
10.1021/JA01054A045
Studies on polyoxins, antifungal antibiotics. 13. The structure of polyoxins.
K. Isono (1969)
10.1021/ol202276h
Diastereoselective control of intramolecular aza-Michael reactions using achiral catalysts.
Cheng Zhong (2011)
10.1016/S0960-894X(99)00064-5
Synthesis of α-C(1→3)-mannopyranoside of N-acetylgalactosamine, a new β-galactosidase inhibitor
C. Pasquarello (1999)
10.1021/JM050968B
Orthogonal activation of the reengineered A3 adenosine receptor (neoceptor) using tailored nucleoside agonists.
Z. Gao (2006)
10.1002/CBER.19550880205
Synthese der D‐Glucosaminuronsäure (2‐Amino‐2‐desoxy‐D‐glucuronsäure) und einige ihrer Derivate (IX. Mitteil. über Oxydative Umwandlungen an Kohlenhydraten)
K. Heyns (1955)
10.1055/S-0029-1216935
Enantioselective Access to All-trans 5-Alkylpiperidine-3,4-diols: Application tothe Asymmetric Synthesis of the 1-N-Iminosugar(+)-Isofagomine
A. Rives (2009)
10.1021/OL049146J
Stereoselective iodocyclization of 3-acylamino-2-methylene alkanoates: synthesis of analogues of N-benzoyl-syn-phenylisoserine.
R. Galeazzi (2004)
10.1002/CHIN.199426243
Synthesis of C-Glycosides of N-Acetylglucosamine by Direct Alkylation of 2-Amino-2-deoxy-2,3,4,6-tetra-O-acetyl Glucopyranosyl Chloride.
Kyung-Il Kim (1994)
Novel antifungal b-amino acids: synthesis and activity against Candida albicans
J Mittendorf (2003)
10.1093/nass/nrn170
Towards fluorous-phase synthesis of nucleoside beta-peptides.
R. Threlfall (2008)
10.1002/CBER.19681011120
Diaminozucker, IX. Synthese der 3‐Amino‐3‐desoxy‐ und 3.6‐Diamino‐3.6‐didesoxy‐D‐glucose
W. M. Z. Reckendorf (1968)
10.3390/M596
Synthesis of rac-tert-butyl 3-(benzyloxycarbonylamino)-2-(4-bromophenyl)-tetrahydrofuran-3-carboxylate
Andreas A Grauer (2009)
10.1055/S-0028-1087545
Synthesis of Unnatural C-2 Amino Acid Nucleosides Using NIS-Mediated Ring Opening of 1,2-Cyclopropane Carboxylated Sugar Derivatives
S. D. Haveli (2009)
10.1248/CPB.42.1251
Synthesis of Nucleosides and Related Compounds. XXXIV. Synthesis of 5-Isonitroso-1, 3-dioxane-4, 6-diones and Their Reactions
Nobuya Katagiri (1994)
Synthesis and stereochemistry of some 1,2,3,4-tetrasubstituted pyrrolidines. Recueil Des Travaux Chimiques Des Pays-Bas
Gp Rozing (1981)
10.1139/V62-343
SYNTHESIS OF DIPEPTIDES CONTAINING 1-AMINOCYCLOALKYLCARBOXYLIC ACIDS: PART II
Patrice Tailleur (1962)
10.1021/CR000045I
beta-Peptides: from structure to function.
R. I. Cheng (2001)
10.1111/J.1399-3011.2004.00143.X
Conformational properties of hybrid peptides containing alpha- and omega-amino acids.
R. Roy (2004)
10.1002/CHIN.200237206
Stereoselective Cycloadditions of Chiral Acyl-Nitroso Compounds; Selective Reactions of Ring-Cleaved Cycloadducts Leading to a New Approach to Polyoxamic Acid.
Adrian G. Pepper (2002)
10.1016/S0040-4020(97)00364-5
Ring opening of sialyllactones with glycine esters: Synthesis of selectively protected glycinyl-NeuAc saccharopeptides
J. Gervay (1997)
10.1021/CR9903003
Methods for anomeric carbon-linked and fused sugar amino Acid synthesis: the gateway to artificial glycopeptides.
A. Dondoni (2000)
10.1016/J.TET.2009.01.108
Synthesis of 5-substituted-3,4-dihydroxycyanopyrrolidines. An easy access to polyhydroxyprolines
Marina Moura (2009)
[The components of the microbial preparation of lysoamidase from the Pseudomonodaceae family responsible for its bacteriolytic activity].
I. Kulaev (1989)
10.1002/1099-0690(200107)2001:13<2547::AID-EJOC2547>3.0.CO;2-H
Preparation and Biological Evaluation of Pyrrolidinediols and Pyrrolidine N-Oxides from D-Ribose Using the Nitrone Approach
A. Palmer (2001)
10.1021/JM00172A036
Synthesis and activity of a potent N-methyl-D-aspartic acid agonist, trans-1-aminocyclobutane-1,3-dicarboxylic acid, and related phosphonic and carboxylic acids.
R. Allan (1990)
10.1248/CPB.24.2312
Azabicycloalkanes as analgetics. V. 4-Phenyl-2-azabicyclo[2,2,2]octanes.
M. Takeda (1977)
10.1002/EJOC.201200103
A Nitro Sugar‐Mediated Stereocontrolled Synthesis of β2‐Amino Acids: Synthesis of a Polyhydroxylated trans‐2‐Amino­cyclohexanecarboxylic Acid
José M Otero (2012)
10.1021/jo800356q
Concise synthesis of (S)-N-BOC-2-hydroxymethylmorpholine and (S)-N-BOC-morpholine-2-carboxylic acid.
K. Henegar (2008)
10.1016/S0008-6215(00)83463-1
9-[3-acetamido-3-C-(carboxymethyl)-3-deoxy-32,2-lactone-α (andβ)-D-xylofuranosyl]adenine-analogs of the nucleoside moiety of the polyoxins
A. Rosenthal (1978)
10.1007/S00706-005-0369-9
Synthesis and Stereostructure of 3-Amino-5- and -6-hydroxybicyclo[2.2.1]heptane-2-carboxylic Acid Diastereomers
M. Palkó (2005)
10.1248/CPB.42.2653
EXPLANATION FOR STEREOSELECTIVITY OF THS CIS-DIHYDROXYLATION OF CIS-3,5-DISUBSTITUTED CYCLOPENTENES
Nobuya Katagiri (1994)
10.1021/OL053144X
Electroreductive intramolecular coupling of aromatic imino esters: is four-membered cyclization much more favorable than six-membered cyclization?
N. Kise (2006)
10.1002/CHIN.200151197
Cyclic Homooligomers from Sugar Amino Acids: Synthesis, Conformational Analysis, and Significance.
E. Locardi (2001)
10.1002/(SICI)1099-0690(200005)2000:9<1745::AID-EJOC1745>3.0.CO;2-8
Sialyltransferase Inhibitors Based on CMP-Quinic Acid
Christoph Schaub (2000)
10.1002/(SICI)1099-0690(199912)1999:12<3483::AID-EJOC3483>3.0.CO;2-E
Regio‐ and Stereoselective Opening of Oxiranes through Neighbouring Group Participation: Stereocontrolled Synthesis of Enantiopure Hydroxylated Oxazolidin‐2‐ones
N. Langlois (1999)
Carbohydr Res
10.1105/tpc.112.103564
Pipecolic Acid, an Endogenous Mediator of Defense Amplification and Priming, Is a Critical Regulator of Inducible Plant Immunity[W]
Hana Návarová (2012)
A compendium of cyclic sugar amino acids 687
10.1021/jo901892d
Synthesis of conformationally constrained diaminodicarboxylic acid derivatives.
Robin A Weatherhead (2009)
10.1002/CHIN.199627225
Mimics of L-Rhamnose: Synthesis of C-Glycosides of L-Rhamnofuranose and an α-Azidoester as Divergent Intermediates for Combinatorial Generation of Rhamnofuranose Libraries.
J. Estévez (1996)
10.1016/j.bmcl.2008.10.101
Oxadiazolone bioisosteres of pregabalin and gabapentin.
D. Wustrow (2009)
10.7164/ANTIBIOTICS.41.1711
Nucleoside antibiotics: structure, biological activity, and biosynthesis.
K. Isono (1988)
Novel helical foldamers
A Ghorai (2010)
10.1016/S0040-4039(01)01676-8
An enantio- and stereocontrolled route to epopromycin B via cinchona alkaloid-catalyzed Baylis-Hillman reaction
Y. Iwabuchi (2001)
10.1016/J.TETASY.2006.06.025
Stereospecific microbial reduction of ethyl 1-benzyl-3-oxo-piperidine-4-carboxylate
Zhiwei Guo (2006)
10.1021/JA9816685
Folded conformation in peptides containing furanoid sugar amino acids
T. Chakraborty (1998)
10.1016/J.TETLET.2012.01.033
Simple conversion of fully protected amino acids to zwitterions
J. Hao (2012)
10.1016/S0040-4020(01)87887-X
Total, Asymmetric-Synthesis of Deoxypolyoxin-C
Y. Auberson (1990)
10.1055/S-2002-19326
Synthesis of α,α-Disubstituted β-Amino Esters and Peptide Derivatives
E. Alonso (2002)
10.1021/JO991399G
Glucose-derived 3'-(carboxymethyl)-3'-deoxyribonucleosides and 2', 3'-lactones as synthetic precursors for amide-linked oligonucleotide analogues.
M. J. Robins (2000)
10.1016/S0040-4039(03)01415-1
Templated scaffolds of cis- and trans-tetrahydrofuran γ-amino acids: γ-azido-β-hydroxy-tetrahydrofuran-2-carboxylates from pentono-δ-lactones
G. J. Sanjayan (2003)
Azidolysis of alpha,beta-epoxycarboxylic acids. A water-promoted process efficiently catalyzed by indium trichloride at pH 4.0.
F. Fringuelli (2001)
10.1002/ARDP.19933260509
Amino Acids, XIV; (±)‐Pipecolic Acid Derivatives, IV: An Efficient Synthetic Method for the Preparation of (±)‐Baikiain and its Derivatives
C. Herdeis (1993)
10.1002/EJOC.201001159
A Cascade Annulation Based Convergent Approach to Racemic Tetrodotoxin
Fernando Cagide-Fagín (2010)
10.1002/CHIN.197927362
SYNTHESIS OF 9-DEOXY-9-ETHOXYCARBONYL-9-AZAPROSTAGLANDIN E2 ETHYL ESTER
G. P. Rozing (1979)
10.1002/1521-3773(20000804)39:15<2761::AID-ANIE2761>3.0.CO;2-9
Carbohydrate Derivatives for Use in Drug Design: Cyclicαv-Selective RGD Peptides
E. Lohof (2000)
10.1002/1521-3765(20021004)8:19<4365::AID-CHEM4365>3.0.CO;2-U
Design, synthesis, and NMR structure of linear and cyclic oligomers containing novel furanoid sugar amino acids.
S. Gruner (2002)
10.1016/J.TETASY.2011.09.021
Stereodivergent approach to both syn- and anti-isomers of γ-amino-β-hydroxy acids: (3S,4S)- and (3R,4S)-AHPPA derivatives
D. Yoo (2011)
10.1002/PRAC.19251110122
Über die Einwirkung schwefligsaurer Salze auf aromatische Amino- und Hydroxylverbindungen. 12. Mitteilung: Über die Produkte der Einwirkung von Sulfiten auf 1,8-Dinitronaphthalin
H. T. Bucherer (1925)
10.1002/anie.201004646
Proof of the existence of an unstable amino acid: pleurocybellaziridine in Pleurocybella porrigens.
T. Wakimoto (2011)
10.1016/S0040-4039(99)00413-X
SYNTHESIS AND BIOLOGICAL ACTIVITY OF DYSIHERBAINE MODEL COMPOUND
M. Sasaki (1999)
10.1016/S0040-4020(03)00049-8
An unusual bicyclic aziridine, 1-azabicyclo[4.1.0]heptan-2-one, and its reaction with nucleophiles
X. Wu (2003)
10.1002/CHIN.200037130
Diastereoselective Synthesis of Hydantoin- and Isoxazoline-Substituted Dispirocyclobutanoids.
K. Park (2000)
10.1021/jo801993k
Stereoselective formation of a functionalized dipeptide isostere by zinc carbenoid-mediated chain extension.
W. Lin (2009)
10.1016/S0040-4039(01)02367-X
Cyclic trimer of 5-(aminomethyl)-2-furancarboxylic acid as a novel synthetic receptor for carboxylate recognition
T. Chakraborty (2002)
10.1055/S-2004-820021
An expeditious route towards pyranopyran sugar amino acids
Gijsbert M. Grotenbreg (2004)
10.1002/CHIN.201012185
An Efficient Route to Acyclic C-Nucleosides and Fused-Ring Analogues of Uridine from exo-Glycals.
Gérald Enderlin (2010)
10.1002/CHIN.199632250
Synthesis of a Potent Inhibitor of β-Glucuronidase.
Y. Igarashi (1996)
10.1111/j.1747-0285.2010.00954.x
The Remarkable Stability of Chimeric, Sialic Acid‐derived α/δ‐Peptides in Human Blood Plasma
Jonel P. Saludes (2010)
10.1016/J.TET.2005.09.037
1-C-(2′-Oxoalkyl) glycosides as latent α,β-unsaturated conjugates. Synthesis of aza-C-glycosides by an intramolecular hetero-Michael addition
T. Yi (2005)
10.1039/B303249N
Synthesis and functional studies of THF-gramicidin hybrid ion channels.
A. Vescovi (2003)
10.1002/chin.198241338
CHEMISTRY OF THE NEOPOLYOXINS, PYRIMIDINE AND IMIDAZOLINE NUCLEOSIDE PEPTIDE ANTIBIOTICS
M. Uramoto (1982)
10.1016/S0008-6215(02)00487-1
Synthesis of new sugar amino acid derivatives of D-glucosamine.
J. Xie (2003)
10.1016/S0960-894X(99)00033-5
Synthesis of a tetrasubstituted bicyclo [2.2.2] octane as a potential inhibitor of influenza virus sialidase.
P. W. Smith (1999)
10.1016/J.TETLET.2009.02.125
An improved synthesis of a fluorescent gabapentin-choline conjugate for single molecule detection.
H. Wu (2009)
10.1055/S-2005-869866
Stereoselective Synthesis of the Conformationally Constrained Glutamate Analogue, (-)-(2R,3S)-cis-2-Carboxyazetidine-3-acetic Acid, from (S)-N-Tosyl-2-phenylglycine
A. Burtoloso (2005)
10.1021/OL0255918
ChemInform Abstract: Synthesis of Different Chiral Amino γ-Butyrolactones and Amino γ-Butenolides.
J. M. Concellón (2002)
10.1093/glycob/cwp039
The CMP-legionaminic acid pathway in Campylobacter: biosynthesis involving novel GDP-linked precursors.
Ian C. Schoenhofen (2009)
10.1016/0040-4039(95)01732-W
Spirodiketopiperazines at the anomeric position of mannopyranose: Novel N- linked glycopeptides incorporating an α- amino acid at the anomeric position of mannopyranose
J. Estévez (1995)
10.1016/J.TETASY.2009.04.010
Stereoselective synthesis of 2-azetidinylglycine and aminopyrrolidone derivatives from Garner’s aldehyde
Latibuddin Thander (2009)
10.1016/J.TETASY.2010.08.013
Enantiospecific synthesis of the sugar amino acid (2S,5S)-5-(aminomethyl)-tetrahydrofuran-2-carboxylic acid
M. L. Uhrig (2010)
10.1002/CHIN.199714161
Synthesis and Biology of the Rigidified Glutamate Analogue, trans-2- Carboxyazetidine-3-acetic Acid (t-CAA).
A. Kozikowski (1996)
10.1002/CHIN.199532201
A New Asymmetric Synthesis of α‐Methylcysteines via Chiral Aziridines.
H. Shao (1995)
10.1002/JLAC.1990199001216
Structural variations of N‐acetylneuraminic acid, 18. Synthesis of the side chain stereo and deoxy analogs of 5‐acetamido‐2,6‐anhydro‐3,5‐dideoxy‐D‐erythro‐L‐manno‐nononic acid
B. Bandgar (1990)
10.1016/S0957-4166(02)00158-1
Synthesis of enantiopure analogues of 3-hydroxyproline and derivatives
A. Avenoza (2002)
10.1016/S0040-4020(01)90479-X
Deoxyiminoalditols from aldonolactones. III. Preparation of 1,4-dideoxy-1,4-imino-L-gulitol. - Evaluation of 1,4-dideoxy-1,4-iminohexitols as glycosidase inhibitors
I. Lundt (1994)
10.1021/JO010299J
Synthesis of a bicyclic analogue of AZT restricted in an unusual O4'-endo conformation.
M. H. Sørensen (2001)
10.1021/JO00362A027
Rapid and convenient syntheses of polyoxin peptides containing N-methylated peptide bonds
J. Boehm (1986)
10.1021/jm050142
Structure-based design, synthesis, and memapsin 2 (BACE) inhibitory activity of carbocyclic and heterocyclic peptidomimetics.
S. Hanessian (2005)
10.1016/S0957-4166(98)00206-7
Spirodiketopiperazines of mannofuranose: carbopeptoid α-amino acid esters at the anomeric position of mannofuranose
J. Estévez (1998)
10.1021/OL034927Q
Oxazolinyloxiranyllithium-mediated stereoselective synthesis of alpha-epoxy-beta-amino acids.
R. Luisi (2003)
10.1002/EJOC.200500062
Facile Regio‐ and Diastereoselective Syntheses of Hydroxylated2‐Aminocyclohexanecarboxylic Acids
F. Fülöp (2005)
10.1021/JO026161Y
Directed dihydroxylation of cyclic allylic alcohols and trichloroacetamides using OsO4/TMEDA.
T. Donohoe (2002)
10.1002/chem.200801826
Stereochemical assignment and first synthesis of the core of miharamycin antibiotics.
F. Marcelo (2008)
10.1002/CHIN.199601227
Enantioselective Total Syntheses of (‐)‐allo‐Coronamic Acid, (‐)‐(Z)‐2, 3‐Methanohomoserine, and (2S,3R)‐Cbz‐cyclo‐Asp‐OMe.
J. Jiménez (1996)
10.1071/CH04014
The Synthesis of Some Oligopeptides Derived from Novel Carbohydrate α-Amino Acids
A. Scaffidi (2004)
10.1016/S0040-4039(97)00496-6
High throughput on-bead monitoring of solid phase reactions by Diffuse Reflectance Infrared Fourier Transform Spectroscopy (DRIFTS)
T. Y. Chan (1997)
10.1071/CH9841123
Synthesis of analogues of GABA. XII. cis- and trans-4-Aminotetrahydrofuran-2-carboxylic acid
R. Allan (1984)
10.1002/1521-3765(20020902)8:17<3976::AID-CHEM3976>3.0.CO;2-7
Synthesis and conformational analysis of fructose-derived scaffolds: molecular diversity from a single molecule.
L. Cipolla (2002)
10.2174/0929867023370941
Sugar amino acids and their uses in designing bioactive molecules.
T. Chakraborty (2002)
10.1016/J.TETASY.2009.02.014
Iodine-mediated ring-closing iodoamination with concomitant N-debenzylation for the asymmetric synthesis of polyhydroxylated pyrrolidines
S. Davies (2009)
10.1016/j.bmcl.2009.03.140
Discovery and structure-activity relationships of pentanedioic acid diamides as potent inhibitors of 11beta-hydroxysteroid dehydrogenase type I.
D. Roche (2009)
10.1016/J.TETASY.2003.12.008
Synthesis of enantiopure 7-azanorbornane proline–α-amino acid chimeras by highly efficient HPLC resolution of a phenylalanine analogue
A. Gil (2004)
10.1002/CHIN.199237240
Preparation of Bicyclic Boroxazolidones from Aziridine-2-carboxylic Esters.
J. Legters (1992)
N: S-acetals
10.1016/J.TETLET.2010.03.051
Flexible palladium-catalysed amidation reactions for the synthesis of complex aryl amides
Christopher W. Barfoot (2010)
10.1002/CHIN.199813183
Solution Phase Synthesis of Amide‐Linked N‐Acetyl Neuraminic Acid, α‐Amino Acid, and Sugar Amino Acid Conjugates.
P. S. Ramamoorthy (1998)
10.1021/JO0605593
Total synthesis and biological evaluation of neodysiherbaine A and analogues.
M. Shoji (2006)
10.1016/J.TET.2004.06.060
Stereoselective synthesis of constrained oxacyclic hydroxyethylene isosteres of aspartyl protease inhibitors. Nitroaldol methodology toward 2,3-substituted tetrahydrofurans
S. Hanessian (2004)
10.1002/PSC.622
The synthesis of oligomers of oxetane‐based dipeptide isosteres derived from L‐rhamnose or D‐xylose
Stephen W. Johnson (2005)
10.1002/PRAC.19080770133
Über die Einwirkung schwefligsaurer Salze auf aromatische Amino‐ und Hydroxylverbindungen
H. T. Bucherer (1908)
10.1080/07328309408009176
Synthesis of a 4-Amino-4-deoxy-D-galacturonic Acid Derivative
Christian Vogel (1994)
10.1039/B612058J
Formation of left-handed helices in hybrid peptide oligomers with cis beta-sugar amino acid and L-Ala as building blocks.
B. Jagadeesh (2007)
10.1021/JM00184A017
(+/-)-trans-2-(Aminomethyl)cyclobutanecarboxylic acid hydrochloride: a rigid analogue of gamma-aminobutyric acid.
J. O'donnell (1980)
10.1016/S0040-4039(00)91559-4
Enantioselective synthesis of loracarbef from sodium erythorbate
Jeffery W. Frazier (1992)
10.1021/ja808286x
Synthesis and structural characterization of sialic acid-glutamic acid hybrid foldamers as conformational surrogates of alpha-2,8-linked polysialic acid.
Jonel P. Saludes (2009)
10.1002/(SICI)1099-0690(200005)2000:9<1831::AID-EJOC1831>3.0.CO;2-S
Deoxyhydantocidin: Synthesis by Base-Catalyzed Spiro Cyclization and Interconversion with the 1′-Epimer
Annabelle Renard (2000)
A Stereospecific Synthesis of (+)-2-Epideoxymannojirimycin and (2R,3R,4R,5R)-3,4,5-Trihydroxypipecolic Acid
박기훈 (1995)
10.1039/B610858J
Self-assembly of cyclic homo- and hetero-β-peptides with cis- furanoid sugar amino acid and β-hGly as building blocks
B. Jagannadh (2006)
10.1016/S0968-0896(02)00033-0
Cytotoxic T lymphocyte epitope analogues containing cis- or trans-4-aminocyclohexanecarboxylic acid residues.
M. Marastoni (2002)
10.1021/JO00364A015
Methyl 2,3-dideoxy-3-nitro-D-erythro-pentofuranoside, isomers and derivatives
J. Weber (1986)
Synthesis of 1-(5-amino-3,5
Min J-M (1999)
10.1016/J.TETASY.2008.11.019
Parallel kinetic resolution of tert -butyl ( RS )-6-alkyl-cyclohex-1-ene-carboxylates for the asymmetric synthesis of 6-alkyl-substituted cishexacin derivatives
S. Davies (2008)
10.1002/CHIN.199517237
The Synthesis of 7-Carbonyl Homologues of 1-Deoxynojirimycin.
A. Kilonda (1995)
Helv Chim Acta
10.1039/B500223K
Cyclic beta-amino acid derivatives: synthesis via lithium amide promoted tandem asymmetric conjugate addition-cyclisation reactions.
S. Davies (2005)
10.1016/J.TETASY.2009.03.009
Pyranocyclopropanyl sugar amino acids, a new class of constrained (di)peptide isosteres
Martijn D. P. Risseeuw (2009)
10.1016/J.TETLET.2004.06.130
Metal-assisted synthesis of enantiopure spirocyclic β-lactams from azetidine-2,3-diones
Benito Alcaide (2004)
10.3998/ARK.5550190.0010.B09
A new entry into 3-hydroxypyrrolidine derivatives from protected α- or β-amino esters
J. Aurrecoechea (2009)
10.1021/JM049927Q
Design, synthesis, and evaluation of sugar amino acid based inhibitors of protein prenyl transferases PFT and PGGT-1.
Farid El Oualid (2004)
10.1021/JA026250S
Design and synthesis of a novel class of sugar-peptide hybrids: C-linked glyco beta-amino acids through a stereoselective "acetate" Mannich reaction as the key strategic element.
C. Palomo (2002)
10.1021/ja300624j
Evidence for helical structure in a tetramer of α2-8 sialic acid: unveiling a structural antigen.
Marcos D. Battistel (2012)
10.1016/S0040-4039(01)80452-4
Cleavage of a nucleosidic oxetane with carbanions: synthesis of a highly promising candidate for anti-HIV agents — a phosphonate isostere of AZT 5′-phosphate
H. Tanaka (1989)
10.1002/EJOC.200300031
Synthesis and Structural Analysis of Cyclic Oligomers Consisting of Furanoid and Pyranoid ϵ-Sugar Amino Acids
R. V. Well (2003)
10.1002/ANIE.200462595
Orthogonally protected sugar diamino acids as building blocks for linear and branched oligosaccharide mimetics.
Frank Sicherl (2005)
10.1016/S0040-4020(01)90035-3
Synthesis of deoxymannojirimycin fagomine deoxynojirimycin 2-acetamido-1,5-imino-1,2,5-trideoxy-D-mannitol 2-acetamido-1,5-imino-1,2,5-trideoxy-D-glucitol 2S,3R,4R,5R-trihydroxypipecolic acid and 2S,3R,4R,5S-trihydroxypipecolic acid from methyl 3-O-benzyl-2,6-dideoxy-2,6-imino-α-D-mannofuranoside
G. Fleet (1987)
10.1021/ja305900r
Poly-amido-saccharides: synthesis via anionic polymerization of a β-lactam sugar monomer.
Eric L Dane (2012)
10.1002/1099-0690(200209)2002:17<2948::AID-EJOC2948>3.0.CO;2-E
Enantiomerically Pure β‐Amino Acids: A Convenient Access to Both Enantiomers of trans‐2‐Aminocyclohexanecarboxylic Acid
A. Berkessel (2002)
10.1073/PNAS.0602537103
Structural insights into stereochemical inversion by diaminopimelate epimerase: an antibacterial drug target.
B. Pillai (2006)
10.1002/CHIN.199743115
Intramolecular O‐H Insertion Reaction of Azido Substituted Diazoesters and Its Relevance to the Mechanism of the Allylic Azide Rearrangement.
A. Pawda (2010)
10.1002/tcr.20144
Diversity-oriented synthesis.
R. J. Spandl (2008)
10.1021/JO702116C
Rapid and efficient synthesis of dysiherbaine and analogues to explore structure-activity relationships.
M. Sasaki (2008)
10.1021/jo9012817
Three-component assembly of amines, boronic acids, and a polyfunctionalized furanose: a concise entry to furanose-based carbohydrate templates.
A. Gómez (2009)
10.1016/J.TET.2010.04.110
Monomers for preparation of amide linked RNA: Synthesis of C3'-homologated nucleoside amino acids from d-xylose.
P. Tanui (2010)
10.1002/CHIN.200006210
Synthesis of Enantiomerically Pure Amino Acids Containing 2,5‐Disubstituted THF Rings in the Molecular Backbone.
A. Schrey (2000)
10.1002/CBDV.200490087
The World of β‐ and γ‐Peptides Comprised of Homologated Proteinogenic Amino Acids and Other Components
D. Seebach (2004)
10.1016/S0957-4166(00)82381-2
Attempted ring contraction of α-triflates of 3-azido- and 3-fluoro-γ-lactones to oxetanes
R. Elliott (1990)
10.1016/J.TETASY.2010.04.051
Constrained cycloalkyl analogues of glutamic acid: stereocontrolled synthesis of (+)-2-aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid (LY354740) and its 6-phosphonic acid analogue
J. Krysiak (2010)
Noninvasive Imaging of αvβ3 Integrin Expression Using 18F-labeled RGD-containing Glycopeptide and Positron Emission Tomography
R. Haubner (2001)
10.1039/c1ob05952a
Amphiphilic allylation of arylidene-1,3-oxazol-5(4H)-one using bis-π-allylpalladium complexes: an approach to synthesis of cyclohexyl and cyclohexenyl α-amino acids.
Afaf R. Genady (2011)
10.1021/ol1010246
Diastereoselective intramolecular additions of allyl- and propargylsilanes to iminium ions: synthesis of cyclic and bicyclic quaternary amino acids.
S. Fustero (2010)
10.1002/PSC.759
Cyclic oligomers of oxetane‐based dipeptide isosteres derived from L‐rhamnose
G. Fleet (2006)
10.1002/CHIN.198948113
Catalytic Cyclopropanation of Alkenes with Ethyl Nitrodiazoacetate. A Facile Synthesis of Ethyl 1-Nitrocyclopropanecarboxylates.
P. E. O'bannon (1989)
10.1002/EJOC.200600228
The Synthesis of cis- and trans-Fused Bicyclic Sugar Amino Acids
Martijn D. P. Risseeuw (2006)
10.1016/S0040-4039(99)01205-8
Conformationally locked nucleosides. Synthesis and stereochemical assignments of 3′-N,5′-C-bridged 3′-amino-3′-deoxythymidines
Guangyi Wang (1999)
10.1016/J.TET.2011.11.023
4-(1-Haloalkyl)-3-nitrotetrahydrofurans as versatile scaffolds for the synthesis of diversely functionalized tetrahydrofurans
U. Jahn (2012)
10.1016/0040-4039(88)85133-5
Acetal-initiated cyclization of allylsilanes to highly functionalized piperidine derivatives
A. Mann (1988)
10.1002/CHIN.199518270
Stereocontrolled Synthesis of Spirodihydrouracil Nucleoside.
H. Sano (1995)
10.1002/CHIN.200306109
Synthesis of Chiral Bicyclic Azetidine Derivatives.
A. Barrett (2003)
10.1016/J.TETASY.2006.06.048
Asymmetric synthesis of pent-3-yl (R)-6-methyl-cyclohex-1-ene carboxylate
N. M. Garrido (2006)
10.1016/S0008-6215(00)85873-5
Selective ring-opening of 3,4,5-tri-O-acetyl-2,6-anhydro-d-glycero-l-manno-heptaric anhydride with ammonia: the synthesis of 7-amino-2,6-anhydro-7-deoxy-l-glycero-l-galacto-heptonic acid
E. Fuchs (1975)
10.1021/jm800792b
A beta-fluoroamine inhibitor of purine nucleoside phosphorylase.
Jennifer M. Mason (2008)
10.1021/jo901277a
Theoretical and experimental studies on alpha/epsilon-hybrid peptides: design of a 14/12-helix from peptides with alternating (S)-C-linked carbo-epsilon-amino acid [(S)-epsilon-Caa((x))] and L-ala.
G. V. M. Sharma (2009)
10.1248/YAKUSHI1947.81.8_1189
Studies on the Synthesis of 1-Deoxy-1-ureidoglucuronic Acid and Related Compounds. V: Synthesis and Infrared Absorption Spectra of 1-Azido-1-deoxy-β-D-glucopyranuronic Acid Derivatives and Methyl 1-Amino-1-deoxy-2, 3, 4-tri-O-acetyl-β-D-glucopyranuronate@@@1-Azido-1-deoxy-β-D-glucopyranuronic Acid誘導
M. Kuranari (1961)
10.1016/0040-4039(96)00327-9
Synthesis of sulfated β-1,6-linked oligosaccharide mimetics: A novel potent inhibitor of HIV replication
Y. Suhara (1996)
10.1021/BM060415Y
Columnar Assembly of Cyclic β-Amino Acid Functionalized with Pyranose Rings
F. Fujimura (2006)
10.1016/j.bmcl.2010.09.067
A new insight on the hypochlorous acid scavenging mechanism of tryptamine and tryptophan derivatives.
L. C. Carvalho (2010)
10.2174/157017808784872160
Synthesis of Sugar β-Amino Acid Containing Homooligomeric Cyclic Peptides
M. Andreini (2008)
10.1021/ja907233q
Stereospecific synthesis of conformationally constrained gamma-amino acids: new foldamer building blocks that support helical secondary structure.
Li Guo (2009)
10.1021/jm100959g
Identification of selective norbornane-type aspartate analogue inhibitors of the glutamate transporter 1 (GLT-1) from the chemical universe generated database (GDB).
Erika Luethi (2010)
10.1021/JO00201A018
dl-Isoserine and related compounds
T. Williams (1985)
10.1021/JM00045A013
Inhibitors of HIV-1 proteinase containing 2-heterosubstituted 4-amino-3-hydroxy-5-phenylpentanoic acid: synthesis, enzyme inhibition, and antiviral activity.
D. Scholz (1994)
10.1039/c2ob26992a
Synthesis of cyclically constrained sugar derived α/β- and α/γ-peptides.
A. Franconetti (2013)
10.1038/nrd1823
Automated synthesis of oligosaccharides as a basis for drug discovery
P. Seeberger (2005)
A compendium of cyclic sugar amino acids 683
10.1002/CHIN.199616238
Novel Oligosaccharide Mimetics by Solid-Phase Synthesis.
C. Mueller (1996)
10.1002/ANIE.199527121
Saccharide–Peptide Hybrids as Novel Oligosaccharide Mimetics†
H. Wessel (1996)
10.1021/jm101156y
Pipecolic acid derivatives as small-molecule inhibitors of the Legionella MIP protein.
Christina Juli (2011)
10.1002/ANIE.200460293
An efficient total synthesis of optically active tetrodotoxin.
T. Nishikawa (2004)
10.3390/ECSOC-14-00381
Synthesis of Conformationally Restricted Glycoamino Acids using Fluorinating Agents
F. Cabrera-Escribano (2010)
10.1016/S0040-4039(00)01693-2
Parallel synthesis of cyclic sugar amino acid:amino acid hybrid molecules
R. V. Well (2000)
10.1071/CH06392
Structural Characterization of a Pentapeptide Derived from a Novel Carbohydrate α-Amino Acid
A. Scaffidi (2007)
Columnar assembly of cyclic beta-amino acid functionalized with pyranose rings.
F. Fujimura (2006)
10.1016/0008-6215(94)84114-4
Acylating properties of N-substituted 2-C:1-N-carbonyl-2-deoxyglycopyranosylamines
D. Mostowicz (1994)
10.1002/CHIN.201218056
Catalytic [3 + 2] Annulation of Aminocyclopropanes for the Enantiospecific Synthesis of Cyclopentylamines.
F. Nanteuil (2012)
Synthesis of 9-azap- rostaglandin analogs
Gp Rozing (1976)
10.1021/JO034586U
Cyclic homooligomers of furanoid sugar amino acids.
T. Chakraborty (2003)
10.1107/S1600536805043205
Pentafluorophenyl (3R,4R,5R)-5-{[(3R,4R,5R)-5-azidomethyl-3,4-dimethoxy-2,3,4,5-tetrahydrofuran-3-carbonylamino]methyl}-3,4-dimethoxy-2,3,4,5-tetrahydrofuran-3-carboxylate
F. Punzo (2006)
J Org Chem
10.3998/ARK.5550190.0006.B18
A convenient synthesis of trans -3-hydroxy-L-proline
S. Sinha (2005)
10.1016/J.TETLET.2005.04.094
Stereoselective synthesis of the various isomers of 3,4-dideoxy furanoid sugar amino acids with methyl substitution at the C6 position
T. Chakraborty (2005)
10.1016/J.BMC.2004.11.044
Exploring human adenosine A3 receptor complementarity and activity for adenosine analogues modified in the ribose and purine moiety.
Philippe van Rompaey (2005)
10.1039/b902366f
Synthesis of pyrrolidine homoazasugars and 3,4-dihydroxy-5-hydroxymethylprolines using aldol additions of metalated bislactim ethers to 2,4-O-ethylidene-D-erythroses.
O. Blanco (2009)
10.1002/CHIN.200435279
Conformational Properties of Hybrid Peptides Containing α‐ and ω‐Amino Acids
R. Roy (2004)
10.1039/B707707F
A new diastereoselective aza-allyl conjugate addition-Michael addition-ring closure reaction sequence and its application in the construction of six contiguous stereogenic centres.
Magdaline Koutsaplis (2007)
10.1007/s00726-011-0894-2
α/β-Peptide foldamers: state of the art
Ludwig K. A. Pilsl (2011)
10.1016/S0968-0896(02)00020-2
Oligomers of glycamino acid.
Y. Suhara (2002)
10.1002/CHIN.199740321
Unnatural Oligomers and Unnatural Oligomer Libraries
M. J. Soth (1997)
10.1016/0006-291X(90)91469-9
Substitution of proline with pipecolic acid at the scissile bond converts a peptide substrate of HIV proteinase into a selective inhibitor.
T. Copeland (1990)
10.1080/07328319708006215
THE SYNTHESIS OF 2'-C-FUNCTIONALISED NUCLEOSIDES FOR INCORPORATION INTO CATALYTIC RNA
A. J. Lawrence (1997)
10.1016/S0040-4039(01)00661-X
10-Helical conformations in oxetane β-amino acid hexamers
T. Claridge (2001)
10.1002/CHIN.199749108
C3-Thia and C3-Carba Isosteres of a Carbocyclic Influenza Neuraminidase Inhibitor, (3R,4R,5S)-4-Acetamido-5-amino-3-propoxy-1- cyclohexene-1-carboxylic Acid.
W. Lew (1997)
A compendium of cyclic sugar amino acids 681
10.1246/CL.1979.819
Synthesis of optically active 4-amino-2-(hydroxymethyl)tetrahydrofuran-4-carboxylic acids.
YoshimuraJuji (1979)
10.7164/ANTIBIOTICS.37.1324
Oxetin, a new antimetabolite from an actinomycete. Fermentation, isolation, structure and biological activity.
S. O̅mura (1984)
10.1016/S0040-4039(00)89000-0
Probing the topography of kainate recognition sites: Synthesis of a novel oxetane containing kainic acid analogue.
A. Kozikowski (1990)
10.1016/S0960-894X(97)00332-6
C3-Thia and C3-carba isosteres of a carbocyclic influenza neuraminidase inhibitor, (3R,4R,5S)-4-acetamido-5-amino-3-propoxyl-1-cyclohexene-1-carboxylic acid
W. Lew (1997)
10.1107/S1600536804022494
(2S,3R,4R,5S)-3,4-O-Iso­propyl­idene-2-methyl-1-oxa-6,9-diaza­spiro[4.5]decane-7,10-dione
D. Watkin (2004)
10.1016/S0040-4039(98)00393-1
Diastereoselective peracid epoxidation: Control of the face selectivity via functional group tuning and proper choice of epoxidation reagent
A. Jensen (1998)
10.1246/CL.1982.1975
A FACILE SYNTHETIC APPROACH TO THE FRAGMENT D OF ANTIBIOTIC NOSIHEPTIDE, 2-[1-AMINO-3-CARBOXY-3-HYDROXY-(1S,3S)-PROPYL]-THIAZOLE-4-CARBOXYLIC ACID
M. Iwakawa (1982)
10.1016/S0040-4039(02)02696-5
Synthesis of the four diastereoisomers of 3-thymine-1-(tbutoxycarbonyl)aminocyclopentane-1-carboxylic acid
N. Howarth (2003)
10.1016/S0040-4039(01)00501-9
Synthesis of a potent (±)-4-(2-hydroxyphenyl) analogue of the acromelic acids by dearomatising cyclisation of a lithiated N-p-methoxybenzyl-4-methoxy-1-naphthamide
A. Ahmed (2001)
10.1021/ja000817s
Total Synthesis of (−)-Dysiherbaine
Hidekazu Masaki (2000)
10.1111/J.1399-3011.2005.00275.X
Furanoid sugar amino acids as dipeptide mimics in design of analogs of vasoactive intestinal peptide receptor binding inhibitor.
S. Prasad (2005)
10.1002/CHIN.200013158
Synthesis of 1-Amino-4-hydroxycyclohexane-1-carboxylic Acids.
A. Avenoza (2000)
10.1016/S0040-4020(02)00158-8
Furanoid sugar amino acid based peptidomimetics: well-defined solution conformations to gel-like structures
T. Chakraborty (2002)
10.1186/1475-2859-8-61
Selectively improving nikkomycin Z production by blocking the imidazolone biosynthetic pathway of nikkomycin X and uracil feeding in Streptomyces ansochromogenes
Guojian Liao (2009)
10.1016/J.TETLET.2011.01.013
Rapid access to cis-cyclobutane γ-amino acids in enantiomerically pure form
Virginie André (2011)
10.1016/J.TET.2008.03.068
Stereoselective synthesis of hydroxylated β-aminocyclohexanecarboxylic acids
Loránd Kiss (2008)
10.1002/PSC.597
Principles of carbopeptoid folding: a molecular dynamics simulation study
Riccardo Baron (2005)
10.1021/JM050169T
Synthetic iminosugar derivatives as new potential immunosuppressive agents.
Xin-Shan Ye (2005)
10.1590/S0103-50531999000300012
Rhodium(II)-Catalysed Intramolecular O-H Insertion of alpha-Diazo-gamma-Azido-delta-Hydroxy-beta-Ketoesters: Evidence for a Novel Sigmatropic Rearrangement of an Allylic Azide Intermediate
A. Padwa (1999)
Synthesis of a, a-disubstituted b-amino esters and peptide derivatives
E Alonso (2002)
10.1016/S0960-894X(01)80254-7
Replacement of the phosphodiester linkage in oligonucleotides: Comparison of two structural amide isomers
A. D. Mesmaeker (1994)
10.1016/J.TETLET.2010.03.083
The design of efficient and selective routes to a key 1,4-cis-substituted cyclohexylamide intermediate
Christopher W. Barfoot (2010)
10.1002/CHIN.200116055
Azidomercurations of Alkenes: Mercury‐Promoted Schmidt Reactions.
W. Pearson (2001)
10.1016/S0040-4039(01)91235-3
Structure and total synthesis of chryscandin, a new antifungal antibiotic
M. Yamashita (1984)
10.1016/j.jmb.2008.10.072
Crystal structure of diaminopimelate epimerase from Arabidopsis thaliana, an amino acid racemase critical for L-lysine biosynthesis.
B. Pillai (2009)
10.1016/S0957-4166(98)00365-6
Intermediates for incorporation of tetrahydroxypipecolic acid analogues of α- and β-d-mannopyranose into combinatorial libraries: unexpected nanomolar-range hexosaminidase inhibitors. Synthesis of α- and β-homomannojirimycin
John P. Shilvock (1998)
10.1021/jm300256z
Cytotoxic effects of combination of oxidosqualene cyclase inhibitors with atorvastatin in human cancer cells.
Davide Staedler (2012)
10.1071/CH06137
An Expansion of the Role of the Corey–Link Reaction for the Synthesis of α-Substituted Carboxylic Acid Esters
A. Scaffidi (2006)
10.1002/EJOC.201100452
Iminosugar Analogues of Phosphatidyl Inositol as Potential Inhibitors of Protein Kinase B (Akt)
Alexandre Orsato (2011)
10.1246/BCSJ.43.246
Synthesis of Cyclic α-Amino Acids. IV. Syntheses of Adenine Nucleosides of 3-Amino-3- C -carboxy-3-deoxy- D -ribofuranose and 3-Amino-3- C -carboxy-3-deoxy- D -ribopyranose
H. Yanagisawa (1970)
10.1002/CHIN.199852238
Ru(II)‐Catalyzed Ring Closing Metathesis in Stereoselective Syntheses of Constrained Homoserine Analogues.
K. Hammer (1998)
10.1016/S0040-4039(97)00138-X
Solution phase synthesis of (1→5)-amide linked sugar amino acid dimers derived from sialic acids
J. Gervay (1997)
10.1002/chin.197844136
A NEW APPROACH TO THE SYNTHESIS OF PRIMARY AMINES, ISOTHIOCYANATES, AND 1-AMINOALKANEPHOSPHONATES VIA N-PHOSPHINYL ALDOXIMES AND KETOXIMES
B. Krzyżanowska (1978)
A compendium of cyclic sugar amino acids 667
10.1016/S0008-6215(99)00057-9
Synthesis of 1-(5-amino-3,5-dideoxy-3-methoxycarbonylmethyl-β-d-ribofuranosyl)thymine
D. Lu (1999)
Synthesis and evaluation of novel 8,6-fused bicyclic peptidomimetic compounds as interleukin-1beta converting enzyme inhibitors.
Steven V O'neil (2005)
10.1007/BF02708268
Sugar amino acids and related molecules: Some recent developments
T. Chakraborty (2004)
10.1039/c1cc10643k
"Inosaminoacids": novel inositol-amino acid hybrid structures accessed by microbial arene oxidation.
Sarah Pilgrim (2011)
10.1039/b719631h
Regioselective intramolecular ring closure of 2-amino-6-bromo-2,6-dideoxyhexono-1,4-lactones to 5- or 6-membered iminuronic acid analogues: synthesis of 1-deoxymannojirimycin and 2,5-dideoxy-2,5-imino-D-glucitol.
B. M. Malle (2008)
10.1021/JM00326A021
THE CHEMISTRY AND PHARMACOLOGY OF A SERIES OF CYCLOALKANESPIRO-5'-HYDANTOINS.
W. Oldfield (1965)
10.1002/CHIN.199939170
Application of 2,3‐Aziridino‐γ‐lactone Methodology Toward the Enantiospecific Synthesis of the (3S,4S)‐Isomer of Dihydroxy‐L‐glutamic Acid.
Philippe Dauban (1999)
10.1039/c0ob00042f
Concise syntheses of selective inhibitors against α-1,3-galactosyltransferase.
G. Zhang (2010)
10.1016/J.TETLET.2004.03.181
Ring-closing alkyne metathesis mediated synthesis of cyclic beta-turn mimetics
M. Ijsselstijn (2004)
10.1021/JO00070A050
Chirospecific synthesis of (1S,3R)-1-amino-3-(hydroxymethyl)cyclopentane, a precursor for carbocyclic nucleoside synthesis. Intramolecular aziridine cyclizations
S. Bergmeier (1993)
10.1080/07328300903261562
Synthesis of 3-Fluoro-Oxetane δ-Amino Acids
S. D. Lucas (2009)
10.1016/S0040-4020(01)87766-8
Behaviour of the gem-cyano-ethoxycarbonyl cyclohexane, thiopyran and pyran derivatives with sodium borohydride and lithium aluminium hydride
F. González (1990)
10.1016/S0040-4039(00)94268-0
A total synthesis of 6-methoxy-epi PS-5 from aminomalonate.
Takeo Yoshioka (1986)
10.1248/CPB.34.3102
Synthesis of a new amino acid-antibiotic, oxetin and its three stereoisomers.
Y. Kawahata (1986)
10.1016/0040-4039(96)00768-X
Studies directed towards the synthesis of miharamycin B
S. Czernecki (1996)
10.1107/S1600536811017764
(2R,6S)-tert-Butyl 2-(benzhydrylcarbamoyl)-6-methylmorpholine-4-carboxylate
H. Wang (2011)
10.1002/CHIN.197049143
HETEROCYCLISCHE BETA-ENAMINOESTER 3. MITT. NMR-SPEKTROSKOPISCHE UNTERSUCHUNGEN DER PROTONIERUNG HETEROCYCLISCHER BETA-ENAMINOESTER
H. Wamhoff (1970)
10.1016/J.TET.2006.05.067
A novel series of oligomers from 4-aminomethyl-tetrahydrofuran-2-carboxylates with 2,4-cis and 2,4-trans stereochemistry
A. A. Edwards (2006)
10.1039/A708555I
Amphiphilic poly(sugar amino acid)s: a novel class of glycoclusters for supramolecular materials
S. Nishimura (1998)
10.1021/JO00084A037
Stereoselective Epoxidation of Phe-Gly and Phe-Phe Vinyl Isosteres
Annika Jenmalm (1994)
10.1021/JO0487449
A practical synthesis of gramicidin s and sugar amino Acid containing analogues.
Gijsbert M. Grotenbreg (2004)
10.1016/J.TET.2012.01.079
Helical secondary structures in 2:1 and 1:2 α/γ-peptide foldamers
L. Guo (2012)
10.1002/CHIN.200235070
ChemInform Abstract: Stereoselective Synthesis of Functionalized γ-Amino Esters: Azetidinium Salts and Epoxy Esters.
J. Concellon (2002)
10.1016/S0040-4039(00)73389-2
The synthesis of cyclobutanol-containing dipeptide analogues
P. Yuan (1994)
10.1021/ol202002r
Three-component coupling approach to trachyspic acid.
Daniel C Schmitt (2011)
10.1016/S0008-6215(00)85132-0
Synthesis of an analog of the nucleoside moiety of the polyoxins
A. Rosenthal (1980)
10.1016/S0040-4020(01)88359-9
Total, asymmetric synthesis of (1r-1-c-(6′-amino-7′h-purin-8′-yl)-1,4-anhydro-3-azido-2,3-dideoxy-d-erythro-pentitol.
V. Jeanneret (1992)
10.1007/s00726-011-0893-3
Foldamers containing γ-amino acid residues or their analogues: structural features and applications
Francelin Bouillère (2011)
Synthesis and local anaesthetic activity of certain basic esters of 1-dialkyl amino cyclohexyl carbinols
MN Aboul-Enein (1991)
10.1016/S0040-4039(99)00110-0
From sequencamers to foldamers? Tetrameric furanose carbopeptoids from cis- and trans-5-aminomethyl-tetrahydrofuran-2-carboxylates
D. D. Long (1999)
10.1002/CHIN.201214227
Mannuronic Acids: Reactivity and Selectivity
Jeroen D. C. Codée (2012)
10.1002/CHIN.199904109
Enantioselective Preparation of (2R)‐ and (2S)‐Azetidine‐2‐carboxylic Acids.
P. Wessig (1999)
10.1002/CHIN.198834333
Synthesis of Racemic 6′β‐Hydroxyaristeromycin (I). A Hydroxycarbocyclic Analogue of Adenosine.
A. B. Cheikh (1988)
10.1021/ja1076102
Diaxial diureido decalins as compact, efficient, and tunable anion transporters.
S. Hussain (2011)
10.1002/PRO.5560070409
The structure of a glycogen phosphorylase glucopyranose spirohydantoin complex at 1.8 Å resolution and 100 K: The role of the water structure and its contribution to binding
M. Gregoriou (1998)
10.1002/CBER.19831160502
Heterocyclische β‐Enaminoester, 30. Darstellung sowie Cycloadditions‐Ringerweiterungs‐Sequenz von Iminophosphoranen heterocyclischer β‐Enaminoester: 6,7‐Dihydrooxepine, ‐thiepine und 3,4‐Dihydro‐2H‐thiocine
H. Wamhoff (1983)
10.1002/0471264180.OR055.01
Synthesis Of Nucleosides
H. Vorbrueggen (2004)
10.1002/CHIN.200140192
Synthesis and Antifolate Evaluation of the Aminopterin Analogue with a Bicyclo[2.2.2]octane Ring in Place of the Benzene Ring.
R. Reynolds (2001)
10.1080/00397919008052870
Synthetic Communication: Synthesis of Optically Pure Analogues of D-Arginine Methyl Ester with Antiarrhythmic Activity
A. Banfi (1990)
10.1021/JA01517A037
The Alkaloids of Tabernanthe iboga. Part VIII1
M. Bartlett (1959)
10.1016/J.TETASY.2003.10.001
Synthesis and transformation of novel cyclic β-amino acid derivatives from (+)-3-carene
Szilvia Gyónfalvi (2003)
10.1016/j.bmcl.2011.09.114
Novel cyclohexyl-amides as potent antibacterials targeting bacterial type IIA topoisomerases.
T. J. Miles (2011)
10.1021/JO0344539
Variable strategy toward carbasugars and relatives. 5.(1) Focus on preparation of chiral nonracemic medium-sized carbocycles.
G. Rassu (2003)
10.1002/CHIN.200802106
A Stereoselective Access to Dihydroxylated Pyrrolidines by Reductive Ring Contraction of 1,2‐Oxazines.
H. Reissig (2008)
10.1016/J.TETLET.2004.05.151
Enantioselective synthesis of (−)-galantinic acid
S. Pandey (2004)
10.2174/0929867003374886
Discovery and development of GS 4104 (oseltamivir): an orally active influenza neuraminidase inhibitor.
W. Lew (2000)
10.1016/J.TETASY.2010.07.018
The formal synthesis of 3-epi jaspine B using stereoselective intramolecular oxa-Michael addition
G. Rao (2010)
Grafting aminocyclopentane carboxylic acids onto the RGD tripeptide sequence generates low nanomolar alphaVbeta3/alphaVbeta5 integrin dual binders.
G. Casiraghi (2005)
10.1016/J.TETLET.2007.06.062
Inter and intramolecular copper(I)-catalyzed 1,3-dipolar cycloaddition of azido-alkynes: synthesis of furanotriazole macrocycles ☆
S. Chandrasekhar (2007)
10.1016/J.TETASY.2008.09.005
The iodolactone approach to enantiopure oxiranes of constrained chiral cyclic β-amino acids
Olivier Songis (2008)
10.1002/CHIN.201020073
Synthesis of 3,4-Fused Bicyclic β-Lactams and Their Transformation into Methyl cis-3-Aminotetrahydrofuran-2-carboxylates.
Erika Leemans (2010)
10.1016/S0040-4020(01)80229-5
2-Acetamido-1,2-dideoxynojirimycin: an improved synthesis
R. Furneaux (1993)
10.1021/JA0670761
Stereochemical diversity in asymmetric cyclization via memory of chirality.
T. Kawabata (2006)
10.3762/bjoc.5.5
Synthesis of new Cα-tetrasubstituted α-amino acids
Andreas A Grauer (2009)
10.1021/JO01273A017
7-Azabicyclo [2.2.1] heptane system. I. Pseudo-4-norcocaine
A. Shafiee (1968)
10.1002/CHIN.200629251
Sugar Amino Acids in Designing New Molecules
T. Chakraborty (2006)
10.1002/chin.198226163
SYNTHESIS OF FOUR STEREOISOMERS OF 4‐AMINO‐2‐(HYDROXYMETHYL)TETRAHYDROFURAN‐4‐CARBOXYLIC ACID
J. Yoshimura (1982)
10.1021/jo00897a051
Heteroatom directed photoarylation. Photochemistry of aryloxyenones
A. Schultz (1975)
10.1055/S-0031-1289767
Asymmetric Synthesis of Pipecolic Acid and Derivatives
A. A. Cant (2012)
10.1002/CHIN.198733320
Synthesis of Deoxymannojirimycin, Fagomine, Deoxynojirimycin, 2-Acetamido-1,5-imino-1,2,5-trideoxy-D-mannitol, 2-Acetamido-1,5-imino-1,2,5-trideoxy-D-glucitol, 2S,3R,4R,5R-Trihydroxypipecolic Acid and 2S,3R,4R,5S-Trihydroxypipecolic A
G. Fleet (1987)
10.1002/CHIN.199833253
Carbohydrate-Based Small-Molecule Scaffolds for the Construction of Universal Pharmacophore Mapping Libraries.
M. Sofia (1998)
10.1107/S1600536805042133
Isopropyl 2,5-anhydro-6-azido-3,6-dide­oxy-d-xylo-hexonate
D. Watkin (2006)
Synthesis of 2-amino-2-deoxy-aD-altrofuranoside derivatives from 2,3-O-isopropylidene-D-glyceraldehyde via bicyclic b-lactam intermediates
M Shiokazi (1989)
10.1016/S0040-4039(99)00944-2
Substrate selectivities of proline hydroxylases
T. Shibasaki (1999)
10.2174/157018008784912117
Structure-Activity Relationship Study of 8-amino-2,8-dideoxy-β -KDO, a Potent CMP-KDO Synthetase Inhibitor
H. Adachi (2008)
10.1039/A805364B
Synthesis of oligomers of tetrahydrofuran amino acids: furanose carbopeptoids
M. Smith (1998)
10.1021/JO050749Y
Stereoselective synthesis of constrained oxacyclic hydroxyethylene isosteres of aspartic protease inhibitors: aldol and Mukaiyama aldol methodologies for branched tetrahydrofuran 2-carboxylic acids.
S. Hanessian (2005)
10.1016/J.TETLET.2004.03.098
A simple acromelic acid analog potentially useful for receptor photoaffinity labeling and biochemical studies
K. Furuta (2004)
10.1039/B111258A
Complex tetrahydrofurans from carbohydrate lactones: THF amino acids as building blocks for unnatural biopolymers
D. D. Long (2002)
10.1002/CHIN.198850183
Acetal-Initiated Cyclization of Allylsilanes to Highly Functionalized Piperidine Derivatives.
A. Mann (1988)
10.1002/CBER.19751080712
Polysaccharidanaloga, I. Synthese von 7‐Amino‐2,6‐anhydro‐7‐desoxy‐D‐glycero‐L‐mannoheptonsäure
E. Fuchs (1975)
10.1002/HLCA.200590175
Differently Glycosidated 2-Amino-2-deoxy-d-glucopyranosiduronic Acids as Building Blocks in Peptide Synthesis†
A. Kyas (2005)
10.1016/J.TETASY.2004.07.031
Oxetane cis- and trans β-amino-acid scaffolds from d-xylose by efficient SN2 reactions in oxetane rings: methyl and hydroxymethyl analogues of the antibiotic oxetin, an oxetane β-amino-acid
Sarah F. Jenkinson (2004)
10.1021/JM950641I
Paracyclophanes: a novel class of water-soluble inhibitors of HIV proteinase.
P. Ettmayer (1996)
10.1016/S0040-4020(01)91497-8
Structures of bulgecins, bacterial metabolites with bulge-inducing activity
S. Shinagawa (1984)
10.1002/CHEM.200500384
An access to 3,4-(aminomethano)proline in racemic and enantiomerically pure form.
Farina Brackmann (2005)
10.1021/jo801156a
Studies directed toward the development of amide-linked RNA mimics: synthesis of the monomeric building blocks.
T. Chakraborty (2008)
10.1016/J.TET.2006.02.007
Synthesis of 4-aminomethyl-tetrahydrofuran-2-carboxylates with 2,4-cis and 2,4-trans relationships
A. A. Edwards (2006)
10.1073/PNAS.95.11.5971
A bait and switch hapten strategy generates catalytic antibodies for phosphodiester hydrolysis.
P. Wentworth (1998)
Noninvasive imaging of alpha(v)beta3 integrin expression using 18F-labeled RGD-containing glycopeptide and positron emission tomography.
R. Haubner (2001)
?)-myriocin. Tetrahedron Asymm
J Gonda (2011)
10.1002/cmdc.200700101
Cis‐Configured Aziridines Are New Pseudo‐Irreversible Dual‐Mode Inhibitors of Candida albicans Secreted Aspartic Protease 2
Björn Degel (2008)
10.1016/S0040-4039(97)00569-8
Synthesis of peptidosialosides and peptidosaccharides
S. Sabesan (1997)
Theoretical and experimental studies on a/e-hybrid peptides: design of a 14/12- helix from peptides with alternating (S)-C-linked carbo-e-amino acid [(S)-epsilon-Caa((x))] and L-ala
Gvm Sharma (2009)
10.1016/J.TET.2006.05.080
Efficient synthesis of carbopeptoid oligomers: insight into mimicry of β-peptide
Y. Suhara (2006)
10.1021/JA035461+
Conformational Analysis of Furanoid ε-Sugar Amino Acid Containing Cyclic Peptides by NMR Spectroscopy, Molecular Dynamics Simulation, and X-ray Crystallography: Evidence for a Novel Turn Structure
Renate Van Well (2003)
3,4,5-Trihydroxy-7-oxa and -7azabicyclo[4.1.0]heptane-2-carboxylic acids: synthesis and evaluation as glycosidase inhibitors
K Ohba (1996)
10.1021/JO982259U
An Enantioselective Ring Expansion Route Leading to Furanose and Pyranose Nucleosides Featuring Spirodiketopiperazines at the Anomeric Position.
L. Paquette (1999)
10.1002/1522-2675(200210)85:10<3455::AID-HLCA3455>3.0.CO;2-#
Synthesis and Biological Evaluation of Protein:Geranylgeranyltransferase I Inhibitors Based on the CaaX Box: Incorporation of Sugar Amino Acids as Dipeptide Isosters
F. E. Oualid (2002)
10.1007/BF00811129
Structural variations of N-Acetylneuraminic acid, 12: A new useful approach to 4-epi- and 8-epi-N-Acetylneuraminic acid
Michael Hartmann (1989)
10.1055/B-003-111719
Synthesis of peptides and peptidomimetics : author, keyword, and preparation index
M. Goodman (2004)
10.1021/JA0588510
Beta-turn modified gramicidin S analogues containing arylated sugar amino acids display antimicrobial and hemolytic activity comparable to the natural product.
Gijsbert M. Grotenbreg (2006)
10.1002/CHIN.200601160
Catalytic Asymmetric Synthesis of Piperidine Derivatives Through the [4 + 2] Annulation of Imines with Allenes.
Ryan P. Wurz (2006)
10.1055/S-2000-6408
A Short and Efficient Synthesis of 2R,3R,4R-3,4-Dihydroxyproline, 1,4-Dideoxy-1,4-imino-l-xylitol, 2R,3R,4R,5S-3,4,5-Trihydroxypipecolic Acid, and 1,5-Dideoxy-1,5-imino-l-iditol
B. Lee (2000)
10.1016/S0040-4020(98)00219-1
Internal activation of acrylate-type dienophiles for the Diels-Alder reaction. Stereoselective synthesis of conformationally constrained glutamate analogs
Y. Ohfune (1998)
10.1016/S0040-4039(99)02187-5
Synthetic studies towards phorboxazole A. Stereoselective synthesis of the C3–C19 bis-oxane oxazole portion of the phorboxazole macrolide
G. Pattenden (2000)
10.1016/S0040-4020(01)81716-6
Polyhydroxylated pyrrolidines from sugar lactomes: Synthesis of 1,4-dideoxy-1,4-imino-d-glucitol from d-galactonolactone and syntheses of 1,4-dideoxy-1,4-imino-d-allitol, 1,4-dideoxy-1,4-imino-d-ribitol, and (2s,3r,4s)-3,4-dihydroxyproline from d-gulonolactone
G. Fleet (1988)
10.1016/J.TET.2005.10.056
Uncatalyzed solventless Diels–Alder reaction of 2-amino-3-nitroacrylate: synthesis of new epimeric 2-amino-3-nitro-norbornene- and norbornane-2-carboxylic acids
Francesco Caputo (2006)
10.1002/CHIR.20248
Classification of conformation for sugar amino acid systems using chiroptical spectroscopy.
A. A. Edwards (2006)
10.1016/S0957-4166(00)86337-5
Synthesis of homochiral β-hydroxy-α-aminoacids [(2S,3R,4R)-3,4-dihydroxyproline and (2S,3R,4R)-3,4-dihydroxypipecolic aicd] and of 1,4-dideoxy-1,4-imino-D-arabinitol [DAB1] and fagomine [1,5-imino-1,2,5-trideoxy-D-arabino-hexitol]
G. Fleet (1990)
Synthesis and biological evaluation of heterocycle containing adamantane 11beta-HSD1 inhibitors.
Vince S. C. Yeh (2006)
10.1002/HLCA.19960790602
C‐Glycoside Analogues of N4‐(2‐Acetamido‐2‐deoxy‐β‐D‐glucopyranosyl)‐L‐asparagine: Synthesis and conformational analysis of a cyclic C‐glycopeptide
M. Hoffmann (1996)
10.1016/S0957-4166(01)00108-2
An efficient route to all eight stereoisomers of a tri-functionalised cyclopentane scaffold for drug discovery
M. Smith (2001)
10.1107/S1600536810039589
(3R,4R,5R)-5-(Acetamidomethyl)-N-benzyl-3,4-dihydroxytetrahydrofuran-3-carboxamide
M. Simone (2010)
10.1016/S0014-827X(00)00016-1
Alicyclic β-amino acids: useful synthons in drug research
F. Fülöp (2000)
10.1021/JO0480040
Helix-forming carbohydrate amino acids.
T. Claridge (2005)
The type-specific substance of Hemophilus influenzae, type d: the natural occurrence of glucosamine uronic acid.
A. R. Williamson (1963)
10.1016/J.TETLET.2008.03.001
Nucleoside derived amino acids (NDA) in foldamer chemistry: synthesis and conformational studies of homooligomers of modified AZT
S. Chandrasekhar (2008)
10.1002/chem.201102902
One-handed helical screw direction of homopeptide foldamer exclusively induced by cyclic α-amino acid side-chain chiral centers.
Yosuke Demizu (2012)
10.1021/JM060917U
Synthesis and metabotropic glutamate receptor activity of S-oxidized variants of (-)-4-amino-2-thiabicyclo-[3.1.0]hexane-4,6-dicarboxylate: identification of potent, selective, and orally bioavailable agonists for mGlu2/3 receptors.
J. Monn (2007)
10.1016/J.BMC.2005.01.033
Synthesis of potent and selective inhibitors of Candida albicans N-myristoyltransferase based on the benzothiazole structure.
K. Yamazaki (2005)
10.1002/CHIN.200451165
The Synthesis of Carbohydrate α-Amino Acids Utilizing the Corey—Link Reaction.
A. Scaffidi (2004)
10.1021/JO00384A060
Palladium-catalyzed denitro-sulfonylation and amination of .beta.,.gamma.-epoxy nitro compounds
R. Tamura (1987)
10.1002/CHIN.200427100
The Three-Component Reaction of Dicarbomethoxycarbene, Aldehydes, and β-Nitrostyrenes: A Stereoselective Synthesis of Substituted Tetrahydrofurans.
V. Nair (2004)
10.1139/V61-165
SYNTHÈSES DE COURTS PEPTIDES RENFERMANT DES ACIDES AMINO-1 CYCLOALKYL CARBOXYLIQUES
Patrice Tailleur (1961)
10.1002/CHIN.200548068
Facile Regio- and Diastereoselective Syntheses of Hydroxylated 2-Aminocyclohexanecarboxylic Acids.
F. Fülöp (2005)
10.1515/znb-2005-1109
Synthese furanoider Zuckeraminos¨auren ausgehend von fermentativ gewonnener 2-Oxo-D-gluconsäure / Synthesis of Furanoid Sugar Amino Acids Starting from Fermentatively Produced 2-Oxo-D-gluconic Acid
S. Schmidt (2005)
10.1016/J.TETASY.2010.01.017
Looking glass inhibitors: scalable syntheses of DNJ, DMDP, and (3R)-3-hydroxy-l-bulgecinine from d-glucuronolactone and of l-DNJ, l-DMDP, and (3S)-3-hydroxy-d-bulgecinine from l-glucuronolactone. DMDP inhibits β-glucosidases and β-galactosidases whereas l-DMDP is a potent and specific inhibitor of α
D. Best (2010)
10.1055/S-1993-25927
Deoxyiminoalditols from Aldonolactones; II. Preparation of 1,4-Dideoxy-1,4-iminohexitols with D- and L-Galacto and D- and L-Ido Configuration: Potential Glycosidase Inhibitors
I. Lundt (1993)
10.1016/S0040-4020(01)90072-9
Systemes bicycliques azotes. Synthese photochimique de 1-azabicyclo [n.2.0]alcanes fonctionnalises
L. Ouazzani-Chadi (1990)
10.1021/OL026126D
Synthesis and NMR studies of cyclopeptides containing a sugar amino Acid.
M. Stoeckle (2002)
Stereoselective synthesis of novel 4,5-epoxy-1,2-oxazin-6-ones and alpha,beta-epoxy-gamma-amino acids from beta-lithiated oxazolinyloxiranes and nitrones.
V. Capriati (2006)
10.1002/chin.198522356
DL-ISOSERINE AND RELATED COMPOUNDS
T. M. Williams (1985)
10.1002/jps.22332
Synthesis and in vitro evaluation of gabapentin prodrugs that target the human apical sodium-dependent bile acid transporter (hASBT).
R. Rais (2011)
10.1002/CHIN.199949251
β‐Peptides: Twisting and Turning
K. Gademann (1999)
Synthese furanoider Zuckeraminosäuren ausgehend von fermentativ gewonnener 2-Oxo-D-gluconsäure
S. Schmidt (2005)
10.1002/CHIN.201010063
Stereospecific Synthesis of Conformationally Constrained γ‐Amino Acids: New Foldamer Building Blocks That Support Helical Secondary Structure.
Li Guo (2010)
10.1021/jo9025258
Cyclobutane amino acid analogues of furanomycin obtained by a formal [2 + 2] cycloaddition strategy promoted by methylaluminoxane.
A. Avenoza (2010)
10.1002/CHIN.199547141
Azetidin-3-ones from (S)-α-Amino Acids and Their Reactions with Nucleophiles: Preparation of Some Azetidine-Containing Amino-Alcohol and Amino-Acid Derivatives.
J. Podlech (1995)
A b-fluoroamine inhibitor of purine nucleoside phosphorylase
Jm Mason (2008)
10.1021/JO971415E
Solid Phase Synthesis and Secondary Structural Studies of (1→5) Amide-Linked Sialooligomers1
L. Szabó (1998)
10.1021/CC9900697
Polymer supported reagents in synthesis: preparation of bicyclo[2.2.2] octane derivates via Tandem Michael addition reactions and subsequent combinatorial decoration.
S. Ley (2000)
Jpn. Kokai Tokkyo Koho
K Nishii (1992)
10.1002/CHIN.200149162
Carbopeptoids: Peptides and Diketopiperazines Incorporating the Anomeric Centre of Mannopyranose.
D. D. Long (2001)
10.1039/c1cc00048a
A general synthetic approach to the amnesic shellfish toxins: total synthesis of (-)-isodomoic acid B, (-)-isodomoic acid E and (-)-isodomoic acid F.
Gilles Lemière (2011)
10.1007/s00726-011-0879-1
Synthesis of new functionalized aziridine-2- and azetidine-3-carboxylic acid derivatives of potential interest for biological and foldameric applications
A. Žukauskaitė (2011)
10.1016/S0040-4039(99)01873-0
Short stereocontrolled synthesis of (2S,3S,4R)-3,4-dihydroxyglutamic acid
N. Langlois (1999)
10.1002/CHIN.201220136
Libraries on Oxetane δ-Amino Acid Scaffolds: Syntheses and Evaluation of Physicochemical and Metabolic Properties.
S. D. Lucas (2012)
10.1016/S0040-4039(96)02314-3
Nucleic acid analog peptide (NAAP). Solid phase synthesis of a DNA analog peptide
M. Fujii (1997)
10.1039/A905771D
Stereoselective synthesis of thymine polyoxin C using an allylic trifluoroacetimidate–trifluoroacetamide rearrangement
A. Chen (1999)
10.1016/0014-5793(95)00612-D
Structure of an acidic polysaccharide present in the bacteriolytic complex lysoamidase
L. M. Likhosherstov (1995)
10.1016/S0957-4166(02)00610-9
Carbocyclic α,β-diamino acids: asymmetric Strecker synthesis of stereomeric 1,2-diaminocyclohexanecarboxylic acids
K. P. Fondekar (2002)
10.1016/S0957-4166(01)00115-X
Synthesis of enantiopure N-protected 4,5-disubstituted 3-pyrrolidinones and N-protected 2,5-disubstituted 3-pyrrolidinones via the Dieckmann reaction of dicarbonyl compounds derived from enantiopure β-amino esters
Yue Wang (2001)
10.1016/S0040-4039(00)74302-4
Oxetane nucleosides with fluorine and azide substitutents: nucleophilic displacements on an oxetane ring
Y. Wang (1991)
10.1016/S0223-5234(01)01230-2
Synthesis and pharmacology of site specific cocaine abuse treatment agents: a new synthetic methodology for methylphenidate analogs based on the Blaise reaction.
H. Deutsch (2001)
10.1016/S0040-4039(00)95023-8
Efficient syntheses of naturally occurring 3,4-dihydroxyprolines: Electrophile-mediated lactonization of 2-amino-3-hydroxy-4-pentenoic acid derivatives
Y. Ohfune (1985)
10.1002/CHIN.199849127
Anionically Induced Decomposition of 2-Ethoxycarbonylprop-2-enyl Peroxides.
Celine Cramay (1998)
10.1016/J.TETLET.2003.08.113
A general and efficient route to enantioselective synthesis of pumiliotoxin A alkaloids via a common key intermediate
B. Wang (2003)
10.1055/S-2007-968002
Synthesis of sugar-lysine chimera with integrated gluco-configured 1,3-hydroxyamine motif
Kaidong Zhang (2007)
10.1021/JO7017137
Diastereoselective synthesis of glutamate-appended oxolane rings: synthesis of (s)-(+)-lycoperdic acid.
J. L. Cohen (2007)
10.1002/CHIN.200632138
Efficient Entry to Diversely Functionalized Spirocyclic Oxindoles from Isatins Through Carbonyl-Addition/Cyclization Reaction Sequences.
Benito Alcaide (2006)
10.1002/CHIN.199415254
Deoxyiminoalditols from Aldonolactones. Part 2. Preparation of 1,4‐ Dideoxy‐1,4‐iminohexitols with D‐ and L‐Galacto and D‐ and L‐Ido Configuration: Potential Glycosidase Inhibitors.
I. Lundt (1994)
10.1016/J.TETLET.2006.02.133
A new strategy for the regio- and stereoselective hydroxylation of trans-2-aminocyclohexenecarboxylic acid
L. Kiss (2006)
10.1002/CHIN.200015247
Sugar Amino Acids and Carbohydrates as Scaffolds and Peptidomimetics
E. Lohof (2010)
10.1021/jm800350u
The structural basis for peptidomimetic inhibition of eukaryotic ribonucleotide reductase: a conformationally flexible pharmacophore.
H. Xu (2008)
10.1016/S0040-4020(01)80952-2
3-amino-2,3-dideoxy-D-erythro-furanose derivatives
M. Cheng (1991)
10.1016/S0040-4039(01)00660-8
cis - and trans -3-Azido-oxetane-2-carboxylate scaffolds: hexamers of oxetane cis -β-amino acids
S. F. Barker (2001)
10.1021/JO00084A005
Synthesis of the Ezomycin Octosyl Nucleoside
S. Knapp (1994)
10.1016/j.bbamem.2010.07.001
Membrane lysis by gramicidin S visualized in red blood cells and giant vesicles.
S. Semrau (2010)
10.7164/ANTIBIOTICS.44.293
Hydantocidin: a new compound with herbicidal activity from Streptomyces hygroscopicus.
M. Nakajima (1991)
10.1002/chin.198243176
SYNTHESIS OF 1-AZIDOCYCLOPROPANECARBOXYLATES FROM 2-AZIDO-2-ALKENOATES
T. Hiyama (1982)
10.1002/ANGE.19860980831
Einfache Synthese von 1‐Amino‐1‐cyclopropancarbonsäuren aus Isocyanessigsäure‐tert‐butylester und Epoxiden; Synthese von 5, 6‐Dihydro‐4H‐1,3‐oxazin‐4‐carbonsäureestern
U. Schoellkopf (1986)
10.1016/J.TET.2005.04.003
Chemistry of domoic acid, isodomoic acids, and their analogues
J. Clayden (2005)
The iodolactone approach to enantiopure oxiranes of constrained chiral cyclic b-amino acids Synthesis of a bicyclic analogue of AZT restricted in an unusual O4 0 -endo conformation
O Songis (2001)
10.1055/S-0029-1218552
Easy Access to ConfigurationallyControlled C-Glycofuranoside-Based BuildingBlocks by Means of Formyl C-Glycofuranosides
Yolanda Vera-Ayoso (2010)
10.1016/S0008-6215(00)87033-0
Preparation of a substituted 3-acetamido-3-deoxy-D-ribofuranosyl bromide suitable for the synthesis of puromycin analogs.
H. S. Khadem (1975)
10.1016/S0040-4020(01)89201-2
Asymmetric synthesis of 34--substituted β-lactams via chiral norephedrine-derived oxazolidines.
S. Cardani (1989)
Novel antifungal b-amino acids: synthesis
W Schönfeld (2003)
10.1016/J.TETASY.2010.09.009
Stereoselective synthesis of pinane-based β- and γ-amino acids via conjugate addition of lithium amides and nitromethane
Zsolt Szakonyi (2010)
10.1080/07328300802061717
Synthesis of 3‐Methoxyoxetane δ‐Amino Acids with D‐lyxo, D‐ribo, and D‐arabino Configurations
S. D. Lucas (2008)
10.1002/CHIN.201149133
TiCl4-Promoted Cyclization Reactions of Aminoacetals and Ethenetricarboxylates Leading to Nitrogen-Containing Heterocycles.
S. Yamazaki (2011)
10.1002/HLCA.19860690617
Synthese von racemischen Aminozuckersäure-lactonen: xylo- und lyxo-2,3-Diacetylamino-5-acetoxypentan-4-olid und -2,3,5-Triacetylaminopentan-4-olid
M. Egli (1986)
10.1002/HLCA.201200436
Ab initio MO Theory – An Important Tool in Foldamer Research: Prediction of Helices in Oligomers of omega-Amino Acids
Carsten Baldauf (2012)
10.1016/J.TET.2008.10.067
Development of two synthetic routes to CE-178,253, a CB1 antagonist for the treatment of obesity
T. A. Brandt (2009)
10.1021/jo0107610
Total synthesis of dysiherbaine.
D. Phillips (2002)
10.1002/CHIN.199931305
Peptides That Contain Unnatural Amino Acids: Toward Artificial Proteins
H. Ishida (1999)
10.1016/S0960-894X(98)00575-7
Design and synthesis of a tetrahydropyran-based inhibitor of mammalian ribonucleotide reductase.
A. Smith (1998)
10.1016/0040-4039(96)00352-8
A general synthesis of oligopeptides containing an oxirane ring in the place of a peptidic bond
A. Mann (1996)
10.1039/JR9600002119
428. Some derivatives of 1-aminocyclopentanecarboxylic acid and related compounds
T. A. Connors (1960)
10.1016/0008-6215(88)84109-0
Somatic antigens of Shigella: structure of the O-specific polysaccharide chain of the Shigella dysenteriae type 7 lipopolysaccharide.
Y. Knirel (1988)
10.1016/j.bmcl.2009.03.024
The discovery of potent, selective, and orally bioavailable PDE9 inhibitors as potential hypoglycemic agents.
M. Deninno (2009)
10.1246/BCSJ.40.431
The synthesis of cyclic amino acids from dialdehydes and nitroacetates.
S. Zen (1967)
10.1016/S0960-894X(98)00231-5
Novel constrained CCK-B dipeptoid antagonists derived from pipecolic acid.
B. Bellier (1998)
10.1039/b810817j
Synthesis and conformational studies of peptides from new C-linked carbo-beta-amino acids (beta-Caas) with anomeric methylamino- and difluorophenyl moieties.
G. V. M. Sharma (2008)
10.3390/M594
Synthesis of (2R,3S)-((1R,2S,5R)-2-isopropyl-5-methylcyclohexyl) 2-(4-bromophenyl)-3-(tert-butoxy-carbonylamino)-tetrahydrofuran-3-carboxylate and (2S,3R)-((1R,2S,5R)-2-isopropyl- 5-methylcyclohexyl)2-(4- bromophenyl)-3-(tert-butoxycarbonylamino)-tetrahydrofuran-3-carboxylate
Andreas A Grauer (2009)
10.1016/J.TETLET.2008.09.069
Hydroxylated C-branched pyrrolidines, C-branched prolines and C-branched piperidines from a 2-C-methyl sugar lactone; efficient azide displacement of a tertiary triflate with inversion of configuration
F. P. Cruz (2008)
10.1021/JO035673P
The three-component reaction of dicarbomethoxycarbene, aldehydes, and beta-nitrostyrenes: a stereoselective synthesis of substituted tetrahydrofurans.
V. Nair (2004)
10.1021/jm9018788
Oxetanes in drug discovery: structural and synthetic insights.
Georg Wuitschik (2010)
10.1016/S0008-6215(00)00099-9
Preparation and structure determination of two sugar amino acids via corresponding hydantoin derivatives.
M. Koóš (2000)
10.1002/EJOC.200200710
Synthesis of Novel Tetrahydropyran‐Based Dipeptide Isosters by Overman Rearrangement of 2,3‐Didehydroglycosides
N. M. Kriek (2003)
10.1246/BCSJ.36.34
Reactions of Alicyclic Aminonitrile
Rokuro Sudo (1963)
10.1021/JO0357216
Variable strategy toward carbasugars and relatives. 6. Diastereoselective synthesis of 2-deoxy-2-amino-5a-carba-beta-L-mannopyranuronic acid and 2-deoxy-2-amino-5a-carba-beta-L-mannopyranose.
G. Rassu (2004)
10.1016/S0040-4039(01)91379-6
The first stereospecific synthesis of (+)-(1r,2s,4r)-4-amino-2-hydroxy-1-cyclopentanemethanol and (+)-carbocyclic thymidine.
L. Oetvoes (1987)
10.1039/c2ob25413a
Enantioselective synthesis of gabapentin analogues via organocatalytic asymmetric Michael addition of α-branched aldehydes to β-nitroacrylates.
Masanori Yoshida (2012)
10.1016/J.BMCL.2004.10.022
Design, synthesis, and structural analysis of inhibitors of influenza neuraminidase containing a 2,3-disubstituted tetrahydrofuran-5-carboxylic acid core.
G. Wang (2005)
10.1007/S10967-009-0059-X
Organic synthesis and biological evaluation of novel “3 + 1” mixed ligands of technetium-99m Gabapentin as receptor imaging agents
A. M. Amin (2010)
10.1073/pnas.1015253108
Creation and manipulation of common functional groups en route to a skeletally diverse chemical library
J. Cui (2011)
10.1016/J.TETLET.2004.12.038
Synthesis of a C3-symmetric macrocycle with alternating sugar amino acid and tyrosine residues
Johan F. Billing (2005)
10.1248/CPB.41.1760
Antiulcer agents. III. Synthesis and antiulcer activity of N-[3-(3-piperidinomethylphenoxy)propyl]pentacyclo[4.2.0.0(2,5).0(3,8).0 (4,7)]-octane carboxamides and related compounds.
T. Hasegawa (1993)
10.1016/J.BMCL.2006.07.055
Synthesis and biological evaluation of heterocycle containing adamantane 11β-HSD1 inhibitors
Vince S. C. Yeh (2006)
10.1016/S0040-4020(99)00405-6
Application of 2,3-aziridino-γ-lactone methodology toward the enantiospecific synthesis of the (3S,4S)-isomer of dihydroxy-L-glutamic acid
Philippe Dauban (1999)
10.1002/chem.201002895
Exploring the conformational and biological versatility of β-turn-modified gramicidin S by using sugar amino acid homologues that vary in ring size.
A. Knijnenburg (2011)
10.1002/CHIN.199748276
Synthesis and Structure-Activity Relationships of Some Novel Oxetane Carbapenems.
Subas M. Sakya (1997)
10.1080/07328300701252623
Transformation of Glucose into a Novel Carbasugar Amino Acid Dipeptide Isostere
Bas Lastdrager (2007)
10.1002/HLCA.19960790402
β‐Peptides: Synthesis by Arndt‐Eistert homologation with concomitant peptide coupling. Structure determination by NMR and CD spectroscopy and by X‐ray crystallography. Helical secondary structure of a β‐hexapeptide in solution and its stability towards pepsin
D. Seebach (1996)
10.1016/S0040-4039(00)61744-6
Cyclic sulphates of δ-lactones in the synthesis of tetrahydrofurans tetrahydropyrans and cyclohexanes
B. M. Skead (1993)
10.1021/JO981310R
Studies of Acyl Nitrene Insertions. A Stereocontrolled Route toward Lankacidin Antibiotics.
D. Williams (1999)
Synthesis and biological
KN Mohana (2012)
10.1002/CHIN.199836350
Carbohydrate-Based Combinatorial Libraries
M. Sofia (1998)
10.1016/S0040-4039(00)88853-X
Inhibition of plant glycosidases by a D-galacturonic acid analog
M. Tong (1990)
10.1016/J.TETLET.2003.10.193
U-4C-3CR versus U-5C-4CR and stereochemical outcomes using suitable bicyclic β-amino acid derivatives as bifunctional components in the Ugi reaction
A. Basso (2004)
10.1021/JO980164M
Carbohydrate-Based Small-Molecule Scaffolds for the Construction of Universal Pharmacophore Mapping Libraries
M. Sofia (1998)
10.1002/HLCA.200390331
Automated Synthesis of Oligosaccharides
E. R. Palmacci (2003)
10.1016/J.TET.2006.02.074
Synthesis of (−)-lentiginosine, its 8a-epimer and dihydroxylated pyrrolizidine alkaloid from d-glucose
Vinod D. Chaudhari (2006)
10.1016/0957-4166(96)00013-4
Mimics of l-rhamnose: Anomeric spirohydantoins and diketopiperazines-approaches to novel N-linked glycopeptides of rhamnofuranose
J. Estévez (1996)
10.1007/BF00761540
Synthesis and testing of the antiviral activity of epoxy and triazo derivatives of cyclohexane
L. A. Mukhamedova (2004)
10.1002/CHIN.200215287
A Field Guide to Foldamers
D. Hill (2002)
10.1002/CHIN.200803235
A Compendium of Sugar Amino Acids (SAA): Scaffolds, Peptide‐ and Glyco‐mimetics
Martijn D. P. Risseeuw (2008)
10.1055/S-1999-3680
Deoxyiminoalditols from Aldonic Acids VI. Preparation of the Four Stereoisomeric 4-Amino-3-hydroxypyrrolidines from Bromodeoxytetronic Acids. Discovery of a New α-Mannosidase Inhibitor
G. Limberg (1999)
10.1016/0040-4039(95)02116-7
Synthesis of uracil polyoxin C from uridine
C. M. Evina (1996)
10.1021/JA9525622
Glycosamino Acids: New Building Blocks for Combinatorial Synthesis
Jason P McDevitt (1996)
10.1016/S0040-4020(03)00288-6
Synthesis of bridged sugar amino acids: a new entry into conformationally locked δ- and ε-amino acids
R. V. Well (2003)
10.1039/B212538B
Optically pure β-substituted β-hydroxy aspartates as glutamate transporter blockers
Johny Wehbe (2003)
10.1093/NASS/NRL087
Synthesis and properties of modified siRNA having amide-linked oligoribonucleosides at their 3' overhang regions.
Reiko Iwase (2006)
10.1021/ol802870c
Total synthesis of FR901483.
C. Carson (2009)
10.1002/CHIN.200642191
A Highly Stereocontrolled Total Synthesis of (—)-Neodysiherbaine A.
K. Takahashi (2006)
10.1002/EJOC.200700677
Asymmetric Diels-Alder Reaction of Aminodienes with a Nonracemic Acrylate Bound to Rink Resin: A Comparison of These Reactions with Their Solution- State Analogues
Olivier Songis (2008)
10.1107/S1600536810038559
Pentafluorophenyl (3R,4R,5S)-5-{[(3R,4R,5S)-5-azidomethyl-3,4-dimethoxy-2,3,4,5-tetrahydrofuran-3-carboxamido]methyl}-3,4-dimethoxy-2,3,4,5-tetrahydrofuran-3-carboxylate
M. Simone (2010)
10.1016/J.BMCL.2007.11.059
α,β-Cyclic-β-benzamido hydroxamic acids: Novel templates for the design, synthesis, and evaluation of selective inhibitors of TNF-α converting enzyme (TACE)
G. Ott (2008)
10.1002/CHIN.199013165
Asymmetric Synthesis of 3,4-cis-Substituted β-Lactams via Chiral Norephedrine-Derived Oxazolidines.
S. Cardani (1990)
10.1016/S0960-894X(97)00395-8
solid phase synthesis of C-terminal carbohydrate modified enkephalins
B. Drouillat (1997)
10.1021/BC034170N
[18F]Galacto-RGD: synthesis, radiolabeling, metabolic stability, and radiation dose estimates.
R. Haubner (2004)
10.1016/S0014-5793(00)01720-8
Structure of the Bordetella pertussis 1414 endotoxin
M. Caroff (2000)
10.1016/J.BMCL.2006.01.088
The synthesis of highly potent, selective, and water-soluble agonists at the human adenosine A3 receptor.
M. Deninno (2006)
10.1016/J.TETASY.2011.02.004
A short stereoselective synthesis of the protected uracil 3'-epi-polyoxin C
J. Gonda (2011)
10.1039/B002996N
Tetrahydrofuran amino acids: Secondary structure in tetrameric and octameric carbopeptoids derived from a D-allo 5-(aminomethyl)tetrahydrofuran-2-carboxylic acid.
N. Hungerford (2000)
10.3762/bjoc.5.1
Reduction of arenediazonium salts by tetrakis(dimethylamino)ethylene (TDAE): Efficient formation of products derived from aryl radicals
M. Mahesh (2009)
10.1016/J.TET.2008.08.001
Stereoselective synthesis of azetidine-derived glutamate and aspartate analogues from chiral azetidin-3-ones
A. Burtoloso (2008)
10.1055/S-2005-871558
Intramolecular nucleophilic epoxidation of γ-amino-α,β-unsaturated esters with an N-hydroperoxymethyl group
D. Yoo (2005)
10.1002/CHIN.199807263
A Short Synthesis of (.+‐.)‐Oxetin.
T. Bach (1998)
10.1002/anie.201103261
Diversity-oriented production of metabolites derived from chorismate and their use in organic synthesis.
J. Bongaerts (2011)
10.1055/S-0030-1258572
A Straightforward Route toNovel α,α-Disubstituted Tetrahydrofuran β-AminoAcids and Spirodiketopiperazines from Sugar Lactones
R. Soengas (2010)
10.1016/j.bmcl.2011.06.084
Conjugate of neamine and 2-deoxystreptamine mimic connected by an amide bond.
Venkatareddy Udumula (2011)
10.1246/BCSJ.49.2511
Aminosugars. XXVI. Synthesis of Amido-bonded Disaccharides Containing Hexosaminuronic Acids
J. Yoshimura (1976)
10.1517/17460441.2011.632002
Peptide and peptoid foldamers in medicinal chemistry
W. Horne (2011)
10.1016/J.TETLET.2007.04.019
Synthesis of 7-azabicyclo[2.2.1]heptane-1,4-dicarboxylic acid, a rigid non-chiral analogue of 2-aminoadipic acid
V. Kubyshkin (2007)
Novel furanoid asubstitued a-amino acid as a potent turn mimic in peptide synthesis
M Martinková (2006)
10.1021/jo8020264
Total synthesis of azumamide E and sugar amino acid-containing analogue.
S. Chandrasekhar (2009)
10.1002/CHIN.200509024
Asymmetric Synthesis of the cis‐ and trans‐Stereoisomers of 4‐Aminopyrrolidine‐3‐carboxylic Acid and 4‐Aminotetrahydrofuran‐3‐carboxylic Acid.
M. E. Bunnage (2005)
10.3987/COM-07-S(W)69
Synthesis of cis-fused pyranopyran and pyranopyridine templates by ring rearrangement metathesis
Alexander Niethe (2007)
10.1021/OL030099P
Synthesis of 4-trifluoromethylated 2-alkyl- and 2,3-dialkyl-substituted azetidines.
J. Jiang (2003)
10.1248/CPB.53.81
Stereospecific synthesis of new 4-amino-1,2,3-cyclohexanetricarboxylic acids and 4-amino-1,3-cyclohexanedicarboxylic acids.
Y. Arakawa (2005)
10.1021/JA0397254
An unusual reverse turn structure adopted by a furanoid sugar amino acid incorporated in gramicidin S.
Gijsbert M. Grotenbreg (2004)
10.1002/CHIN.200302178
Synthesis of Sugar Azido or Amino Esters and Their Use as Building Blocks for the Preparation of Saccharide Nucleosides.
J. Xie (2003)
10.1016/S0957-4166(03)00274-X
Synthesis of polyhydroxylated α-nitrocyclohexane carboxylic acids derived from d-glucose: a striking case of racemization
R. Soengas (2003)
Synthesis of nucleosides Rh(II)-catalyzed intramolecular N-H insertion of D-glucosederived d-amino a-diazo b-ketoester: synthesis of pyrrolidine iminosugars
H Vorbrueggen (1999)
10.7164/ANTIBIOTICS.37.1284
Chryscandin, a novel peptidyl nucleoside antibiotic. II. Structure determination and synthesis.
M. Yamashita (1984)
10.1002/CHIN.200518131
C(6)-Alkylation of 3-Hydroxypiperidine via Reductive and Homolytic Cleavage of N,S-Acetals.
M. Bartels (2005)
10.1016/J.TETLET.2005.06.093
Synthesis of dysiherbaine analogue
M. Shoji (2005)
10.1128/AAC.00443-11
Tripropeptin C Blocks the Lipid Cycle of Cell Wall Biosynthesis by Complex Formation with Undecaprenyl Pyrophosphate †
H. Hashizume (2011)
10.1016/S0040-4039(00)01425-8
Synthesis and structural studies of oligomers of 6-amino-2,5-anhydro-6-deoxy-d-mannonic acid
T. Chakraborty (2000)
Quinolone derivatives
S Seto (2012)
10.1016/J.TET.2009.05.077
An alternative synthesis of Tamiflu®: a synthetic challenge and the identification of a ruthenium-catalyzed dihydroxylation route
K. Yamatsugu (2009)
10.1002/CHIN.200208285
2-Benzyl-3,4-iminobutanoic Acid as Inhibitor of Carboxypeptidase A.
Jeong-il Park (2002)
10.1021/JO0349328
Studies on the synthesis of (2S,3R)-3-hydroxy-3-methylproline via C2-N bond formation.
J. Shen (2003)
10.1111/J.1527-3458.2007.00024.X
The preclinical properties of a novel group II metabotropic glutamate receptor agonist LY379268.
G. Imre (2007)
10.1016/J.BBRC.2003.10.119
Inhibition of human salivary α-amylase by glucopyranosylidene-spiro-thiohydantoin
G. Gyémánt (2003)
Synthesis and tumor inhibiting activity of lanthanum (III) complexes with some 1-aminocycloalkancarboxylic acids.
T. B. Kovachev (1996)
10.1016/J.TETLET.2007.11.178
Rapid access to CF3 -containing heterocycles
A. Dobbs (2008)
10.1002/CHIN.200037225
δ-Peptide Analogues of Pyranosyl-RNA. Part 1. Nucleo-δ-peptides Derived from Conformationally Constrained Nucleo-δ-amino Acids: Preparation of Monomers.
G. Karig (2000)
10.1021/jo900296d
Cross-metathesis reactions as an efficient tool in the synthesis of fluorinated cyclic beta-amino acids.
S. Fustero (2009)
10.1002/JLAC.197819781223
13C-NMR-Untersuchungen an Mutarotationsgemischen C-6- und C-4- sowie C-6-modifizierter Amadoriverbindungen
W. Funcke (1978)
10.1002/HLCA.19870700618
Diasterio‐ und enantioselektive Reduktion von β‐Ketoestern mit Cyclopentanon‐, Cyclohexanon‐, Piperidon‐ und Tetralon‐Struktur durch nicht fermentierende Bäcker‐Hefe
D. Seebach (1987)
10.1016/0040-4039(95)01414-D
exo-2-Phenyl-7-azabicyclo[2.2.1]heptane-1-carboxylic acid: A new constrained proline analogue
A. Avenoza (1995)
10.2174/1386207023330200
Sugar amino acid based scaffolds--novel peptidomimetics and their potential in combinatorial synthesis.
T. Chakraborty (2002)
10.1016/J.TETASY.2004.06.003
Asymmetric Strecker synthesis of enantiopure 2,4-ethanothreonines
U. Meyer (2004)
Fleet GWJ (1994b) Tri- and tetra-peptides incorporating an a-amino
JC Estevez (1994)
A novel type of spironucleosides: 20,50-O-bis-TBDMS uridine-30spiro-30- isoxazolidin-50-one and its thymidine congener. Nucleosides Nucleotides
JMJ Tronchet (2006)
10.1021/ja909874b
Chiral lithium(I) binaphtholate salts for the enantioselective direct Mannich-type reaction with a change of syn/anti and absolute stereochemistry.
M. Hatano (2010)
10.1039/c1ob06279d
Design and synthesis of trans-3-aminopyran-2-carboxylic acid (APyC) and α/β-peptides with 9/11-helix.
G. V. M. Sharma (2011)
10.1016/0040-4039(96)01646-2
Synthesis of 2,6-anhydro-3-deoxy-5-O-phosphono-3-tetradecanamido-4-O-[(R)-3-(tetradecanoyloxy)tetradecanoyl]-d-glycero-d- ido-heptonic acid as a new potent endotoxin antagonist and its dimeric analogue
M. Shiozaki (1996)
10.1039/B006192L
Synthesis of bicyclic sugar azido acids and their incorporation in cyclic peptides
F. Peri (2000)
10.1021/OL0269704
Asymmetric synthesis of the putative structure of (-)-oryzoxymycin.
M. Bunnage (2003)
tols as glycosidase inhibitors
Y Maeda (1996)
10.1039/c1cc11689d
HYDRAmers: design, synthesis and characterization of different generation novel Hydra-like dendrons based on multifunctionalized adamantane.
G. Lamanna (2011)
10.7164/ANTIBIOTICS.38.1182
Structure activity relationships of synthetic antibiotic analogues of chryscandin.
T. Komori (1985)
10.1021/JO025538X
Toward a general strategy for the synthesis of 3,4-dihydroxyprolines from pentose sugars.
C. Taylor (2002)
10.1055/S-1997-5747
Novel Strategies for the Synthesis of Peptides containing Cis- or Trans-β-Aminocyclopropanecarboxylic Acids
C. Bubert (1997)
10.1021/OP010204F
Large-Scale Syntheses of FMOC-Protected Non-Proteogenic Amino Acids: Useful Building Blocks for Combinatorial Libraries
J. Dener (2001)
10.1016/J.TETASY.2003.10.005
Total synthesis of 3,4-dihydroxyprolines, d-threo-l-norvaline and (2S,3R,4R)-2-amino-3,4-dihydroxytetrahydrofuran-2-carboxylic acid methyl ester
R. Soengas (2003)
10.1002/chem.200902332
Backbone regulation mimicry by beta-peptidic foldamers: formation of a 10-helix in a mixed 6-strand/14-helix conformational pool.
B. Jagadeesh (2009)
10.1002/CHIN.201112055
Three-Component Coupling Reactions of Silyl Glyoxylates, Vinyl Grignard Reagent, and Nitroalkenes: An Efficient Highly Diastereoselective Approach to Nitrocyclopentanols.
Gregory R. Boyce (2011)
10.1016/S0040-4039(98)00438-9
A new short synthesis of deoxyhydantocidin derivatives
Annabelle Renard (1998)
10.1016/S0040-4020(01)00129-6
New synthesis of all four 1-amino-2-hydroxycyclohexanecarboxylic acids
A. Avenoza (2001)
10.1002/CHIN.201028245
(Pseudo)amide‐Linked Oligosaccharide Mimetics: Molecular Recognition and Supramolecular Properties
J. Blanco (2010)
10.1016/0040-4020(86)80025-4
The synthesis and antimicrobial activity of (1s,2s)-1-hydroxy-2-[(s)-valylamino]cyclobutane-1-acetic acid (1) and (1s, 2s)-1-hydroxy-2-aminocyclobutane-1-acetic acid (2)
J. Baldwin (1986)
10.1039/B701848G
Strained azetidinium ylides: new reagents for epoxidation.
Audrey Alex (2007)
10.1016/S0957-4166(97)00261-9
Synthesis of and from S-pyroglutamic acid. Regio- and diastereoselective ring opening of its derivatives
C. Herdeis (1997)
10.1016/S0040-4020(01)86061-0
Asymmetric synthesis of functionalized α -amino-β-hydroxy acids via chiral norephedrine-derived oxazolidines
S. Cardani (1988)
Gellman SH (2012a) New preorganized c-amino acids as foldamer building
L Guo (2012)
10.1021/JM980616N
Synthesis, pharmacological characterization, and molecular modeling of heterobicyclic amino acids related to (+)-2-aminobicyclo[3.1.0] hexane-2,6-dicarboxylic acid (LY354740): identification of two new potent, selective, and systemically active agonists for group II metabotropic glutamate receptors.
J. Monn (1999)
Nucleosides Nucleotides
10.1016/J.BMCL.2004.04.036
Conformationally restricted analogs of deoxynegamycin.
B. Raju (2004)
10.1021/JO00023A015
Total synthesis of 6-deoxy-6-aminoheptopyranuronic acid derivatives
Giovanni Casiraghi (1991)
10.1002/BIP.20694
Molecular assembly formation of cyclic hexa-beta-peptide composed of acetylated glycosamino acids.
Tatsuya Hirata (2007)
10.1021/JA0607133
Carbohydrate amino acids: the intrinsic conformational preference for a beta-turn-type structure in a carbopeptoid building block.
R. A. Jockusch (2006)
10.1002/EJOC.200700791
Versatile Synthesis of Free and N‐Benzyloxycarbonyl‐Protected 2,2‐Disubstituted Taurines
Boyuan Wang (2008)
10.1021/JO025897S
Synthesis of 2,4-methanoproline analogues via an addition-intramolecular substitution sequence.
T. Rammeloo (2002)
J Chem Soc, Perkin Trans
10.1002/CHIR.20117
Circular dichroism studies of carbopeptoid-cyclodextrins.
A. A. Edwards (2005)
10.1021/OL062098D
Total synthesis of (-)-5,6,11-trideoxytetrodotoxin and its 4-epimer.
T. Umezawa (2006)
10.1055/S-2007-970743
Rh(II)-Catalyzed Intramolecular N-H Insertion of d-Glucose-Derived δ-Amino α-Diazo β-Ketoester: Synthesis of Pyrrolidine Iminosugars
V. P. Vyavahare (2007)
10.1002/EJOC.200801173
New Concise Route to 2-Amino-3-hydroxycycloalkanecarboxylic Acids by Imidate-Mediated Intramolecular Conjugate Addition
Y. Matsushima (2009)
10.1080/00397919008051475
ANALOGS OF GLUTAMIC ACID : SYNTHESIS AND BIOLOGICAL EVALUATION
G. Kraus (1990)
10.1186/1475-2859-11-135
Novel polyoxins generated by heterologously expressing polyoxin biosynthetic gene cluster in the sanN inactivated mutant of Streptomyces ansochromogenes
Jin'e Li (2012)
10.1002/CHIN.200221286
Carbohydrate-Based Mimetics in Drug Design: Sugar Amino Acids and Carbohydrate Scaffolds
S. Gruner (2002)
10.1055/S-1996-4191
Synthesis of (1’S,3’R)-3-(3’-Amino-2’,2’-dimethylcyclobutyl)propan-1-ol from (-)-β-Pinene
J. Blanco (1996)
10.1016/J.TETASY.2008.09.026
Regio- and stereoselective synthesis of constrained enantiomeric β-amino acid derivatives
Zsolt Szakonyi (2008)
10.1080/00397911.2010.515354
Synthesis and Characterization of Novel Bi- and Tricyclic α-Amino Acids
M. Johnson (2011)
10.1246/BCSJ.79.768
On the Stereoselectivity of Asymmetric Strecker Synthesis in a Cyclohexane System : Synthesis of Optically Active cis- and trans-1-Amino-2-hydroxycyclohexane-1-carboxylic Acids
T. Shinada (2006)
10.1021/ol101078z
Synthesis of 5-azaindoles via a cycloaddition reaction between nitriles and donor-acceptor cyclopropanes.
M. M. A. R. Moustafa (2010)
10.1107/S160053680500067X
2-Azido-2-deoxy-3,4-O-isopropylidene-2-C-methyl-d-talono-1,5-lactone
Sarah F. Jenkinson (2010)
10.1039/c1cc16082f
Quantum confinement controlled photocatalytic water splitting by suspended CdSe nanocrystals.
M. A. Holmes (2012)
10.1007/s00726-011-0849-7
C-3 branched δ-3,5-cis- and trans-THF sugar amino acids: synthesis of the first generation of branched homooligomers
M. I. Simone (2011)
10.1016/j.bmcl.2008.03.050
Design and synthesis of morpholine derivatives. SAR for dual serotonin & noradrenaline reuptake inhibition.
P. V. Fish (2008)
10.1016/J.TETASY.2008.07.036
Efficient and stereoselective synthesis of (2S,3S,4S)-3,4-dihydroxyglutamic acid via intramolecular epoxidation
H. Kim (2008)
10.1021/JA073992I
Synthesis of tamiflu and its phosphonate congeners possessing potent anti-influenza activity.
J. Shie (2007)
10.1080/15257770701490399
Foldamers Derived From Nucleoside β-Amino Acids: Pna Or Dna? Can We Have Both In One Place?
R. Threlfall (2007)
10.1002/(SICI)1099-1387(199910)5:10<425::AID-PSC222>3.0.CO;2-O
Designing secondary structures: 5‐azidomethyl tetrahydrofuran‐2‐carboxylates as carbohydrate‐derived dipeptide isosteres
M. Smith (1999)
10.1002/chin.200649195
Efficient Synthesis of Sugar Iminopyrrolidine Derivatives via an Intramolecular Staudinger—Aza‐Wittig‐Type Reaction.
H. Ducatel (2006)
10.1016/S0040-4039(00)87272-X
Synthesis of 1-azidocyclopropanecarboxylates from 2-azido-2alkenoates
T. Hiyama (1982)
10.1139/V81-205
Lewis acid promoted reactions of ethyl cyanoformate. Reaction with 2,5-dimethylfuran
A. W. Mcculloch (1981)
10.1016/S0040-4039(01)00551-2
Novel and efficient transformation of α-amino nitrile to α-imino and α-amide nitriles in asymmetric Strecker synthesis
K. Namba (2001)
10.1002/CHIN.200903259
β‐Peptidic Peptidomimetics
D. Seebach (2009)
10.1016/0957-4166(96)00067-5
Synthesis of a new enantiomerically pure constrained homoserine
A. Avenoza (1996)
10.1055/S-0031-1289702
Exploiting the Addition of Trimethyl(trifluoromethyl)silaneto Functionalized N-Benzylimines forthe Preparation of Two Novel x-Trifluoromethyl x-Amino Acids
A. Tkachenko (2012)
10.1002/CHIN.198745321
3,6-Dideoxy-3,6-imino-1,2-O-isopropylidene-α-D-glucofuranose as a Divergent Intermediate for the Synthesis of Hydroxylated Pyrrolidines: Synthesis of 1,4-Dideoxy-1,4-imino-L-gulitol, 1,4-Dideoxy-1,4-imino-D-lyxitol, 2S,3S,4R-3,4-Dihyd
G. N. Austin (1987)
10.1002/CHIR.1180
Application of L-threonine aldolase-catalyzed reaction to the preparation of protected 3R,5R-dihydroxy-L-homoproline as a mimetic of idulonic acid.
T. Miura (2001)
10.1021/OL0484106
Metathesis approach to the synthesis of polyheterocyclic structures from oxanorbornenes.
J. Winkler (2004)
10.1002/CHIN.198752369
Structure Elucidation of the Glycopeptide Antibiotic Complex A40926.
J. Waltho (1987)
10.1016/J.TETASY.2008.12.012
Carbon-branched δ-tetrahydrofuran sugar amino acids (SAAs) as dipeptide isostere scaffolds
M. I. Simone (2008)
10.1007/BF00119142
Design of superactive and selective integrin receptor antagonists containing the RGD sequence
H. Kessler (2004)
10.1021/jo035312
Synthesis of oligomers derived from amide-linked neuraminic acid analogues.
Travis Q. Gregar (2004)
10.1002/PSC.488
An unsaturated peptidomimetic assembly derived from a carbohydrate
Y. Chung (2004)
10.1016/J.BMCL.2006.08.082
Design, total synthesis, and biological evaluation of neodysiherbaine A derivative as potential probes.
M. Sasaki (2006)
10.1016/S0040-4020(99)00345-2
Synthesis of optically active N-allyl amino compounds with defined trisubstituted double bonds
U. Bösche (1999)
10.1002/EJOC.200500177
Preparation of Cyclopropane Analogues of the Natural AntibioticTAN 1057 A/B
M. Kordes (2005)
10.1021/ol1003302
Synthesis and structural analysis of a new class of azaspiro[3.3]heptanes as building blocks for medicinal chemistry.
Johannes A. Burkhard (2010)
10.1016/0020-708X(78)90142-4
Synthesis and purification of 11C-carboxyl-labeled amino acids
R. Hayes (1978)
10.1002/chin.198637325
The Synthesis and Antimicrobial Activity of (1S,2S)-1-Hydroxy-2-[(S)-valylamino]cyclobutane-1-acetic Acid and (1S,2S)-1-Hydroxy-2-aminocyclobutane-1-acetic Acid.
J. Baldwin (1986)
10.1080/00397919508012674
Synthesis of Polyhydroxylated 6-N-Benzylpiperidin-2-Ones. A Novel Access to 1, 5-Dideoxy-1, 5-imino-D-xylitol
F. Boyer (1995)
10.1039/A805401K
Secondary structure in oligomers of carbohydrate amino acids
M. Smith (1998)
10.1002/CHIN.200850095
Catalytic Hydrogenation of 5,6‐Dihydro‐4H‐1,2‐oxazines Bearing a Functionalized Methylene Group at C‐3.
A. Sukhorukov (2008)
10.1021/ol201043d
In situ generation of the Coates catalyst: a practical and versatile catalytic system for the carbonylation of meso-epoxides.
P. Ganji (2011)
10.1002/chin.198648321
Synthesis of 2R,3S,4R‐Dihydroxyproline from D‐Ribonolactone.
J. C. Dho (1986)
10.1002/JLCR.956
The synthesis of isotopically labeled (+)‐2‐aminobicyclo[3.1.0]hexane‐2,6‐carboxylic acid and its 2‐oxa‐ and 2‐thia‐analogs
W. J. Wheeler (2005)
10.1002/chem.201101855
Synthesis and structural characterization of homochiral homo-oligomers of parent cis- and trans-furanoid-β-amino acids.
S. Pandey (2011)
10.1021/jm801632a
Toward the back-up of boceprevir (SCH 503034): discovery of new extended P4-capped ketoamide inhibitors of hepatitis C virus NS3 serine protease with improved potency and pharmacokinetic profiles.
S. Bogen (2009)
10.1021/JM00164A058
Renin inhibitors containing isosteric replacements of the amide bond connecting the P3 and P2 sites.
J. S. Kaltenbronn (1990)
10.1021/OP050066K
A Practical Synthesis of the Dual Matrix Metalloprotease/Tumor Necrosis Factor Inhibitor MMP090
J. Slade (2005)
10.1016/S0040-4039(97)01133-7
Intramolecular OH insertion reaction of azido substituted diazoesters and its relevance to the mechanism of the allylic azide rearrangement
A. Padwa (1997)
10.1002/cbic.200800139
Synthesis of Novel DC‐SIGN Ligands with an α‐Fucosylamide Anchor
G. Timpano (2008)
10.1080/15257779908041536
Novel TSAO derivatives modified at positions 3" and 4" of the spiro moiety.
E. Lobatón (1999)
10.1016/J.TET.2010.09.109
Spiranic d-gluco-configured N-substituted thiohydantoins as potential enzymatic inhibitors
C. Gasch (2010)
b-Amino acids: function and synthesis
RP Cheng (2001)
10.1002/(SICI)1522-2675(19981216)81:12<2218::AID-HLCA2218>3.0.CO;2-0
Preparation and Structure ofβ-Peptides Consisting of Geminally Disubstitutedβ2,2- andβ3,3-Amino Acids: A Turn Motif forβ-Peptides
D. Seebach (1998)
10.1002/ANIE.199406871
A Sugar Amino Acid as a Novel Peptidomimetic
E. V. Roedern (1994)
10.1039/C39940000111
Total synthesis of (+)-polyoxin J starting from myo-inositol
N. Chida (1994)
10.1021/JA963290L
β-Peptide Foldamers: Robust Helix Formation in a New Family of β-Amino Acid Oligomers
D. Appella (1996)
10.1021/JO00816A020
Synthesis and gramine alkylation of some 3-piperidones. Synthetic route to 2-(3-indolylmethyl)-4-piperidineacetic acid derivatives
R. Sundberg (1971)
Synthesis of the two enantiomers of the carbocyclic analog of nicotinamide ribose and analysis of their biological properties
M Ikbal (1989)
10.1039/c0cc01724h
Novel helical foldamers: organized heterogeneous backbone folding in 1 : 1 alpha/nucleoside-derived-beta-amino acid sequences.
S. Chandrasekhar (2010)
10.1016/S0957-4166(03)00498-1
Selenium-promoted synthesis of enantiomerically pure substituted morpholines starting from alkenes and chiral aminoalcohols
M. Tiecco (2003)
10.1016/J.TET.2006.01.095
Peracid dependent stereoselectivity and functional group contribution to the stereocontrol of epoxidation of (E)-alkene dipeptide isosteres
Daniel Wiktelius (2006)
10.1021/JO9711246
Solution Phase Synthesis of Amide-Linked N-Acetyl Neuraminic Acid, α-Amino Acid, and Sugar Amino Acid Conjugates1
P. S. Ramamoorthy (1997)
10.1016/S0960-894X(02)01022-3
Solid-phase synthesis of cyclic RGD-furanoid sugar amino acid peptides as integrin inhibitors.
Renate M van Well (2003)
10.1038/363418A0
Rational design of potent sialidase-based inhibitors of influenza virus replication
M. Itzstein (1993)
10.1016/S0957-4166(98)00440-6
Synthesis of an eight carbon homologue of α-homomannojirimycin via a bicyclic aminolactone
John P. Shilvock (1998)
10.1016/s0008-6215(01)00239-7
Syntheses of hydantocidin and C-2-thioxohydantocidin.
M. Shiozaki (2002)
10.1021/JO00311A026
SYNTHESIS OF C(6)-CARBOXYLATE ANALOGUES OF N-ACETYLMURAMIC ACID
S. Hecker (1990)
10.1016/J.TETASY.2008.03.030
Oxetane amino acids: synthesis of tetrameric and hexameric carbopeptoids derived from l-ribo 4-(aminomethyl)-oxetan-2-carboxylic acid
Beatrice Lopez-Ortega (2008)
10.1021/JO01029A004
The Reaction of N-Bromosuccinimide with Bicyclo[2.2.1]-5-heptene-endo-cis-2,3-dicarboxylic Anhydride1
L. Zalkow (1964)
10.1002/EJOC.200500977
A Conformationally Locked Aminomethyl C-Glycoside and Studies on ItsN-Pyren-1-ylcarbonyl Derivative Inserted into Oligodeoxynucleotides
C. Verhagen (2006)
10.1055/S-1996-5375
Nucleophilic Opening of Epoxide by Guanidine. A Route to Potential Substrates or Inhibitors of NO Synthases1
C. Gravier-Pelletier (1996)
A SHORT ROUTE TO ALPHA -CHLORO- AND ALPHA -AZIDO-ULOSONIC ESTERS
M. Lakhrissi (1998)
10.1107/S1600536806012487
cyclo {[(6-Amino-6-deoxy-2,3:4,5-di-O-isopropylidene-D-galactonic acid)-(D-Phe)]2}
Richard Bream (2006)
10.1248/CPB.12.1525
THE ABSOLUTE CONFIGURATION OF OPTICALLY ACTIVE ISOVALINE.
S. Yamada (1964)
10.1039/A902411E
Model studies of the overall 5-endo-trig iodocyclization of homoallylic alcohols
Simon B Bedford (1999)
10.1021/ol203144v
Iron-catalyzed [3 + 2] annulation of aminocyclopropanes with aldehydes: stereoselective synthesis of aminotetrahydrofurans.
F. Benfatti (2012)
10.1002/CHIN.200549259
Carbohydrates as Versatile Platforms in the Construction of Small Compound Libraries
Mattie S. M. Timmer (2005)
10.1002/CHIN.200738037
Highly Diastereoselective Synthesis of vicinal Quaternary and Tertiary Stereocenters Using the Iodo-aldol Cyclization.
Frédèric Douelle (2007)
10.1002/CHIN.200229255
Glycosamino Acids: Building Blocks for Combinatorial Synthesis — Implications for Drug Discovery.
F. Schweizer (2002)
10.1016/S0040-4039(01)80831-5
Synthesis of 2S-carboxy-3R, 4R, 5S-trihydroxypiperidine, a naturally occurring inhibitor of β-D-glucuronidase
R. Bernotas (1985)
10.1002/CHIN.201049144
Synthesis of 5‐Azaindoles via a Cycloaddition Reaction Between Nitriles and Donor—Acceptor Cyclopropanes.
M. M. A. R. Moustafa (2010)
10.1002/CHIN.199536231
Synthesis of the Potent Influenza Neuraminidase Inhibitor 4-Guanidino Neu5Ac2en. X-Ray Molecular Structure of 5-Acetamido-4-amino-2,6- anhydro-3,4,5-trideoxy-D-erythro-L-gluco-nononic Acid.
M. Chandler (1995)
10.1016/j.bmcl.2008.01.075
Potent, exceptionally selective, orally bioavailable inhibitors of TNF-alpha Converting Enzyme (TACE): novel 2-substituted-1H-benzo[d]imidazol-1-yl)methyl)benzamide P1' substituents.
G. Ott (2008)
10.1016/J.TET.2009.03.038
Stereocontrolled synthesis of (5+5), (5+6) and (6+6) 3-spiropseudonucleosides
C. Gasch (2009)
10.1021/jo900842w
Conformationally restricted nonchiral pipecolic acid analogues.
D. Radchenko (2009)
10.1055/S-1997-708
VINYLCYCLOPROPYLACYL RADICALS. INTRAMOLECULAR KETENE ADDITIONS LEADING TO CONCISE SYNTHESES OF CYCLOHEXENONES
Nicola Herbert (2004)
10.1021/JA01189A085
The Hydrogenation of Esters to Alcohols at 25-150°
H. Adkins (1948)
10.1016/S0040-4039(00)79957-6
Synthesis of C-glycosides of N-acetylglucosamine by direct alkylation of 2-amino-2-deoxy-2,3,4,6-tetra-O-acetyl glucopyranosyl chloride
Kyung-Il Kim (1994)
10.1016/J.TETASY.2004.11.058
Synthesis of C6-substituted 3,4-dideoxy furanoid sugar amino acids
T. Chakraborty (2005)
10.1351/pac198153010113
Stereoselective syntheses of branched-chain sugar derivatives
J. Yoshimura (1981)
10.1002/CHIN.200147172
Synthesis of Constrained Prolines by Diels—Alder Reaction Using a Chiral Unsaturated Oxazolone Derived from (R)-Glyceraldehyde as Starting Material.
E. Buñuel (2001)
10.1002/ANIE.198607541
Simple Synthesis of 1‐Amino‐1‐cyclopropanecarboxylic Acids from tert‐Butyl Isocyanoacetate and Epoxides; Synthesis of Alkyl 5,6‐Dihydro‐4H‐1,3‐oxazine‐4‐carboxylates
U. Schoellkopf (1986)
10.1016/J.MOLCATB.2012.03.005
Microbial enantioselective removal of the N-benzyloxycarbonyl amino protecting group
M. Maurs (2012)
A compendium of cyclic sugar amino acids 679
10.1016/S0040-4039(00)84755-3
Enantiospecific syntheses of 2S,3R,4R,5S-trihydroxypipecolic acid, 2R,3R,4R,5S-trihydroxypipecolic acid, 2S,4S,5S-dihydroxypipecolic acid, and bulgecinine from D-glucuronolactone
B. P. Bashyal (1986)
Reynoso-Soto EA, Ochoa-Teran A (2011) Microwaveassisted synthesis of cycloalkanespirohydantoins and piperidinespirohydantoins as precursors of restricted a-amino acids
IA Rivero (2011)
10.1016/S0040-4039(99)00109-4
Absence of secondary structure in a carbopeptoid tetramer of a trans-5-aminomethyl-tetrahydrofuran-2-carboxylate
M. Smith (1999)
10.1002/CHIN.200425128
Fluoropyrrolidine Amides as Dipeptidyl Peptidase IV Inhibitors.
C. Caldwell (2004)
10.1002/ANIE.200501055
C9 Helices and Ribbons in γ‐Peptides: Crystal Structures of Gabapentin Oligomers
P. G. Vasudev (2005)
10.1016/S0040-4039(98)00872-7
A short route to α-chloro- and α-azido-ulosonic esters
M. Lakhrissi (1998)
10.1016/J.BMC.2004.12.035
Synthesis and biological evaluation of lipophilic Ca(1)a(2)L analogues as potential bisubstrate inhibitors of protein:geranylgeranyl transferase-1.
Farid El Oualid (2005)
10.1021/ol8024567
Iodocyclization of chiral CF3-allylmorpholinones: a versatile strategy for the synthesis of enantiopure alpha-Tfm-prolines and alpha-Tfm-dihydroxyprolines.
Caroline Caupène (2009)
10.1128/AAC.00124-10
Damage of the Bacterial Cell Envelope by Antimicrobial Peptides Gramicidin S and PGLa as Revealed by Transmission and Scanning Electron Microscopy
Mareike Hartmann (2010)
10.1016/S0960-894X(98)00267-4
A new series of cyclic amino acids as inhibitors of S-adenosyl L-methionine synthetase.
K. Lavrador (1998)
10.1021/ol801213c
Direct asymmetric intramolecular alkylation of beta-alkoxy-alpha-amino esters via memory of chirality.
K. Moriyama (2008)
10.1016/S0040-4020(96)01180-5
Synthesis of methacrylic-type peroxidic compounds and study of their homolytic induced decomposition in solution
D. Colombani (1997)
10.1016/j.bmc.2010.08.027
Design, synthesis, biological evaluation, and modeling of a non-carbohydrate antagonist of the myelin-associated glycoprotein.
O. Schwardt (2010)
10.3998/ARK.5550190.0012.221
Microwave-assisted synthesis of cycloalkanespirohydantoins and piperidylspirohydantoins as precursors of restricted α-amino acids
I. Rivero (2011)
10.1021/OL048750R
Alkylated sugar amino acids: a new entry toward highly functionalized dipeptide isosters.
Michael Raunkjaer (2004)
10.1016/0040-4020(95)00425-8
Regiochemical control of the ring opening of 1,2-epoxides by means of chelating processes.9. Synthesis and ring opening reactions of cis- and trans-oxides derived from 3-(benzyloxymethyl)cyclopentene and methyl 2-cyclopenten-1-carboxylate 1
M. Colombini (1995)
10.1016/J.TETASY.2004.08.032
Synthesis of enantiopure cis- and trans-2-aminocyclohexane-1-carboxylic acids from octahydroquinazolin-4-ones
J. M. Priego (2004)
10.1055/S-0030-1258498
Solvent-Free and StereoselectiveSynthesis of C-Glycosides by Michael-Type Additionof Enamino Esters to 2-Nitro-d-glucal
T. Zhang (2010)
10.1080/07328303.2011.609627
Libraries on Oxetane δ-Amino Acid Scaffolds: Syntheses and Evaluation of Physicochemical and Metabolic Properties
S. D. Lucas (2011)
Inhibition of human salivary alpha-amylase by glucopyranosylidene-spiro-thiohydantoin.
G. Gyémánt (2003)
10.1016/J.BMCL.2006.09.035
Discovery of potent and selective inhibitors of 11β-HSD1 for the treatment of metabolic syndrome
Steven T. Richards (2006)
10.1039/B705750D
Synthesis of alkylated sugar amino acids: conformationally restricted L-Xaa-L-Ser/Thr mimics.
Martijn D. P. Risseeuw (2007)
10.1016/j.bpj.2012.12.038
Membrane interactions and pore formation by the antimicrobial peptide protegrin.
T. Lazaridis (2013)
J Mol Cat B: Enz
10.1016/0957-4166(96)00012-2
Mimics ofl-rhamnose: Synthesis of C-glycosides of L-rhamnofuranose and an α-azidoester as divergent intermediates for combinatorial generation of rhamnofuranose libraries
J. Estévez (1996)
10.1016/S0957-4166(99)00486-3
Gram-scale synthesis of a glucopyranosylidene-spiro-thiohydantoin and its effect on hepatic glycogen metabolism studied in vitro and in vivo
L. Somsák (2000)
10.1016/J.TETLET.2003.10.103
Huge (14-, 21-, 28-, 35-, 56- and 70-membered ring) macrocyclic lactams––a novel family of carbopeptoid-cyclodextrins
B. Mayes (2004)
10.1002/CHIN.199920177
Deoxyiminoalditols from Aldonic Acids. Part 6. Preparation of the Four Stereoisomeric 4-Amino-3-hydroxypyrrolidines from Bromodeoxytetronic Acids. Discovery of a New α-Mannosidase Inhibitor.
G. Limberg (1999)
10.1002/CHIN.200635214
Synthesis of (‐)‐Lentiginosine (I), Its 8a‐Epimer and Dihydroxylated Pyrrolizidine Alkaloid (II) from D‐Glucose.
Vinod D. Chaudhari (2006)
10.1016/j.bmcl.2010.02.051
Potent ketoamide inhibitors of HCV NS3 protease derived from quaternized P1 groups.
S. Venkatraman (2010)
10.1002/CHIN.200106160
Synthesis and conformational studies of peptidomimetics containing furanoid sugar amino acids and a sugar diacid.
T. Chakraborty (2000)
Jr SR. The alkaloids of tabernanthe iboga. VII. Derivatives of isoquinuclidine
Lh Werner (1958)
10.1016/j.bmc.2011.10.045
Conformationally restricted analogs of the direct thrombin inhibitor FM 19.
E. A. Girnys (2011)
10.1055/S-2000-6267
Enantioselective Synthesis of α,α′-Disubstituted Piperidines via Ruthenium-Catalyzed Ring Rearrangement
U. Voigtmann (2000)
10.1002/CHIN.200039184
A New, Scalable Preparation of a Glucopyranosylidene‐spiro‐thiohydantoin: One of the Best Inhibitors of Glycogen Phosphorylases.
L. Somsák (2000)
10.1016/S0960-894X(02)00958-7
Novel antifungal β-amino acids: synthesis and activity against Candida albicans
J. Mittendorf (2003)
10.1016/j.bmcl.2009.09.083
Preliminary SAR analysis of novel antiproliferative N(6),5'-bis-ureidoadenosine derivatives.
M. Peterson (2009)
10.1002/HLCA.19950780211
Synthesis of Potential Inhibitors of Ethylene Biosynthesis: The diastereoisomers of 1‐amino‐2‐bromocyclopropanecarboxylic acid
L. Wick (1995)
10.1039/b911247m
Alpha,gamma-cyclic peptide ensembles with a hydroxylated cavity.
César Reiriz (2009)
10.1016/0045-2068(90)90037-6
Design and synthesis of potent inhibitors of glutamine synthetase: 1. Cyclic analogs of phosphonothricin
C. Johnson (1990)
10.1002/CHIN.198204203
SYNTHESIS AND STEREOCHEMISTRY OF SOME 1,2,3,4-TETRASUBSTITUTED PYRROLIDINES
G. P. Rozing (1982)
10.1016/S0040-4020(01)92964-3
Heterocyclische β-enaminoester—III
H. Wamhoff (1970)
10.1002/HLCA.19950780510
(±)-4-Amino-4,5-dideoxyribose, (±)-4-amino-4-deoxyerythrose, and (±)-dihydroxyproline derivatives from N-dienyl-γ-lactams
J.‐B. Behr (1995)
10.1016/S0040-4039(99)00697-8
Design and synthesis of a protein:Farnesyltransferase inhibitor based on sugar amino acids
H. Overkleeft (1999)
10.1016/S0040-4020(01)88357-5
Total asymmetric syntheses of d-lividosamine and 2-acetamido-2,3-dideoxy-d-arabino-hexose derivatives. ☆
Etienne de Buchteneere (1992)
10.1016/S0040-4039(01)93129-6
EZOAMINUROIC ACID, 3‐AMINO‐3,4‐DIDEOXY‐D‐XYLO‐HEXAPYRANUROIC ACID, AS A CONSTITUENT OF EZOMYCINS A1 AND A2
K. Sakata (1974)
10.1080/15257770008033851
Conformationally Locked Nucleosides. Synthesis of Oligodeoxynucleotides Containing 3′-Amino-3′-deoxy-3′-N,5′(R)-C-ethylenethymidine
G. Wang (2000)
10.1016/J.TET.2005.09.128
Stereocontrolled synthesis of thiohydantoin spironucleosides from sugar spiroacetals
J. Fuentes (2006)
10.1016/S0040-4039(97)01316-6
Radical cyclisation of amino aldehydes leading to hydroxy pyrrolidines and piperidines
A. Parsons (1997)
10.1016/S0040-4039(98)02089-9
A solid phase approach to oligomers of carbohydrate amino-acids: Secondary structure in a trimeric furanose carbopeptoid
D. D. Long (1998)
10.1016/J.EJMECH.2007.08.010
Novel N-(phosphonomethyl) glycine derivatives: Design, characterization and biological activity.
E. D. Naydenova (2008)
10.1021/jo900966b
Synthesis and solution conformation of homo-beta-peptides consisting of N-mannofuranosyl-3-ulosonic acids.
M. Andreini (2009)
10.1002/CHIN.198739172
Palladium-Catalyzed Denitro-Sulfonylation and Amination of β,γ-Epoxy Nitro Compounds.
R. Tamura (1987)
10.1021/jm800930w
Development of novel G-protein-coupled receptor 54 agonists with resistance to degradation by matrix metalloproteinase.
K. Tomita (2008)
U ¨ ber Tetraamino-adipinsäure und b, b'- Diamino-a, a'-dioxy-adipinsäure
W Traube (1913)
10.1002/CHIN.200347027
Oxazolinyloxiranyllithium‐Mediated Stereoselective Synthesis of α‐Epoxy‐β‐amino Acids.
R. Luisi (2003)
10.1016/J.TETASY.2009.03.004
Stereocontrolled transformation of nitrohexofuranoses into cyclopentylamines via 2-oxabicyclo[2.2.1]heptanes. IV: Synthesis of enantiopure methyl (1S,2R,3R,4R,5S)-5-benzyloxycarbonylamino-2,3-isopropylidenedioxy-4-methoxycyclopentanecarboxylate
F. Fernandez (2009)
Peptide sweeteners
JW Tsang (1984)
10.1021/OL0477529
Convergent approach to (E)-alkene and cyclopropane peptide isosteres.
P. Wipf (2005)
10.1021/JO0502899
Synthesis of orthogonally protected cyclic homooligomers from sugar amino acids.
M. Ménand (2005)
10.7164/ANTIBIOTICS.27.963
Purification and characterization of a sialidase inhibitor, siastatin, produced by Streptomyces.
H. Umezawa (1974)
10.1016/S0960-894X(99)00192-4
Efficient inhibition of muscle and liver glycogen phosphorylases by a new glucopyranosylidene-spiro-thiohydantoin.
E. Ősz (1999)
10.1002/CHIN.199310268
Syntheses of Sialic Acid Isomers with Inhibitory Activity Against Neuraminidase.
T. Yamamoto (1993)
10.1016/j.carres.2011.03.030
Synthesis of 4-amino-4,5-dideoxy-L-lyxofuranose derivatives and their evaluation as fucosidase inhibitors.
Carine Chevrier (2011)
10.1002/chin.198110246
TOTAL SYNTHESIS OF 2,4-METHANOPROLINE
M. C. Pirrung (1981)
10.1016/S0957-4166(99)00205-0
3-Azidotetrahydrofuran-2-carboxylates: monomers for five-ring templated β-amino acid foldamers?
M. Watterson (1999)
10.1016/0040-4039(95)00197-K
POTENT INHIBITION OF GLYCOGEN PHOSPHORYLASE BY A SPIROHYDANTOIN OF GLUCOPYRANOSE : FIRST PYRANOSE ANALOGUES OF HYDANTOCIDIN
C. J. F. Bichard (1995)
10.1016/S0960-894X(98)00153-X
Synthesis of DNA analogues with novel carboxamidomethyl phosphonamide and glycinamide internucleoside linkages.
V. Efimov (1998)
10.1016/J.TETASY.2004.08.023
Pseudoenantiomeric oxetane δ-amino acid scaffolds derived from L-rhamnose and D-xylose: D/L-alanine-D-serine and glycine-L-serine dipeptide isosteres
S. Johnson (2004)
10.1002/CHIN.199814176
C-Glycosides: A Stereoselective Synthesis of α-C-Galactosamines with a Glycosyl Dianion.
F. Burkhart (1998)
10.1016/S0040-4039(01)01845-7
Isothiocyanatoulosonates, a new type of glycosyl isothiocyanate useful for the stereocontrolled synthesis of thiohydantoin spironucleosides
C. Gasch (2001)
10.1055/S-0030-1258464
Synthesis of (±)-8-Oxa-3-azabicyclo[3.2.1]octan-2-thioneand (±)-2-Oxa-5-azabicyclo[2.2.1]heptan-6-thione:Potential Synthons for the Preparation of Novel Heteroaryl-AnnulatedBicyclic Morpholines
Daniel P. Walker (2011)
10.1016/S0040-4020(01)89047-5
Iminoheptitols as glycosidase inhibitors: Synthesis of α-homomannojirimycin, 6-epi-α-homomannojirimycin and of a highly substituted pipecolic acid
I. Bruce (1992)
10.1016/J.TET.2004.11.024
Cyclic peptides containing a δ-sugar amino acid: synthesis and evaluation as artificial receptors
Johan F. Billing (2005)
10.1002/CHIN.200034038
Polymer Supported Reagents in Synthesis: Preparation of Bicyclo[2.2.2]octane Derivatives via Tandem Michael Addition Reactions and Subsequent Combinatorial Decoration.
S. Ley (2000)
10.1002/EJOC.200300805
Synthesis of Imino Sugar Scaffolds for the Generation of Glycosidase Inhibitor Libraries
B. L. Ferla (2004)
10.1002/CHIN.200627267
Recent Advances in Asymmetric Synthesis of Pipecolic Acid and Derivatives
C. Kadouri-Puchot (2006)
10.1016/J.TETASY.2006.07.027
Sugar amino acids at the anomeric position of carbohydrates : synthesis of spirocyclic amino acids of 6-deoxy-L-lyxofuranose
Y. Blériot (2006)



This paper is referenced by
10.1021/acs.joc.5b01049
Orthogonally Protected Furanoid Sugar Diamino Acids for Solid-Phase Synthesis of Oligosaccharide Mimetics.
F. John (2015)
10.1007/s00726-019-02730-5
Isolation from Stevia rebaudiana of DMDP acetic acid, a novel iminosugar amino acid: synthesis and glycosidase inhibition profile of glycine and β-alanine pyrrolidine amino acids
R. F. Martínez (2019)
10.1016/J.TET.2017.10.038
Synthesis and conformational studies of short mixed γ/α-glycopeptides based on sugar γ3,3-amino acids
Mylène Richard (2017)
10.1002/EJOC.201801541
Synthesis of Sulfonimidamide‐Based Amino Acid Building Blocks with Orthogonal Protecting Groups
P. K. Chinthakindi (2019)
10.1039/c5ob00622h
Tetrahydrofuran amino acid-containing gramicidin S analogues with improved biological profiles.
S. Pal (2015)
10.1039/C4RA16196C
An insight into the synthesis of novel aryl-substituted alicyclic β-amino acid derivatives through substrate-directed palladium-catalysed regio- and stereoselective cross-coupling
Melinda Nonn (2015)
10.1002/EJOC.201800943
Synthetic Pathways to 3,4,5-Trihydroxypiperidines from the Chiral Pool
Adam Wood (2018)
10.1016/J.TETASY.2016.08.011
An update on the stereoselective synthesis of γ-amino acids
M. Ordóñez (2016)
10.1016/J.TET.2014.02.063
Stereocontrolled transformation of cyclohexene β-amino esters into syn- or anti-difunctionalized acyclic β2,3-amino acid derivatives
Maria Cherepanova (2014)
10.1007/7081_2015_181
Polyhydroxylated Cyclic Delta Amino Acids: Synthesis and Conformational Influences on Biopolymers
André Wuttke (2015)
10.1039/c3cc48850k
Conformational modulation of peptide secondary structures using β-aminobenzenesulfonic acid.
S. S. Kale (2014)
10.1007/s00726-019-02702-9
α/β-Chimera peptide synthesis with cyclic β-sugar amino acids: the efficient coupling protocol
A. Nagy (2019)
10.1002/tcr.201700038
Selective Synthesis of Fluorine-Containing Cyclic β-Amino Acid Scaffolds.
L. Kiss (2018)
10.1107/S2056989015017582
Crystal structure of 3-C-(N-benzyloxycarbonyl)aminomethyl-3-deoxy-1,2:5,6-di-O-isopropylidene-α-d-allofuranose
Vitālijs Rjabovs (2015)
10.1021/acs.jcim.6b00488
Predictable Conformational Diversity in Foldamers of Sugar Amino Acids
D. Menyhárd (2017)
10.1002/slct.201904430
Solid‐Phase Synthesis of Clickable Psicofuranose Glycocarbamates and Application of Their Self‐Assembled Nanovesicles for Curcumin Encapsulation
M. Vangala (2020)
10.1002/SLCT.201700403
An Insight into Substrate‐Dependent Fluorination of some Highly Substituted Alicyclic Scaffolds
L. Kiss (2017)
10.1016/J.CCLET.2015.04.026
Recent progress of sugar amino acids: Synthetic strategies and applications as glycomimetics and peptidomimetics
Guangzong Tian (2015)
10.1002/chem.201501249
Conformational Plasticity in Glycomimetics: Fluorocarbamethyl-L-idopyranosides Mimic the Intrinsic Dynamic Behaviour of Natural Idose Rings.
Luca Unione (2015)
10.3390/molecules24010161
Alicyclic β- and γ-Amino Acids: Useful Scaffolds for the Stereocontrolled Access to Amino Acid-Based Carbocyclic Nucleoside Analogs
A. Remete (2019)
10.1002/AJOC.201500286
Stereocontrolled Synthesis of Difunctionalized Azetidinones and β2, 3‐Amino Acid Derivatives from Cyclodienes by Ring‐Opening and Cross‐Metathesis Reactions
Márton Kardos (2015)
10.1002/chem.201503998
Benzylidene Acetal Protecting Group as Carboxylic Acid Surrogate: Synthesis of Functionalized Uronic Acids and Sugar Amino Acids.
A. Banerjee (2016)
10.1016/j.tet.2019.130837
Highly functionalized cyclic and bicyclic β−amino acids from sugar β−nitroesters
José M Otero (2020)
10.1002/EJOC.201301705
One-Pot Tandem Strecker Reaction and Iminocyclisations: Syntheses of Trihydroxypiperidine α-Iminonitriles
B. Ayers (2014)
10.1039/C6RA13898E
Construction of quaternary stereocentres on carbohydrate scaffolds
Smritilekha Bera (2016)
10.1021/jo501571j
Asymmetric synthesis of chiral heterocyclic amino acids via the alkylation of the Ni(II) complex of glycine and alkyl halides.
H. Chen (2014)
10.1039/c4ob02421d
Conformational modulation of peptides using β-amino benzenesulfonic acid ((S)Ant).
G. Priya (2015)
10.1002/EJOC.201900101
Chemodiscrimination of Olefin Bonds Through Cross‐Metathesis Reactions – Synthesis of Functionalized β‐Lactam and β‐Amino Acid Derivatives
Melinda Nonn (2019)
10.1021/acs.joc.5b00463
3-Fluoroazetidinecarboxylic Acids and trans,trans-3,4-Difluoroproline as Peptide Scaffolds: Inhibition of Pancreatic Cancer Cell Growth by a Fluoroazetidine Iminosugar.
Zilei Liu (2015)
10.3389/fchem.2015.00040
CNS active O-linked glycopeptides
E. M. Jones (2015)
10.1039/c5ob00668f
Azetidine- and N-carboxylic azetidine-iminosugars as amyloglucosidase inhibitors: synthesis, glycosidase inhibitory activity and molecular docking studies.
Kishor S. Gavale (2015)
10.1016/J.TET.2015.10.001
Glycosylation and functionalization of native amino acids with azido uronic acids
C. J. Cara (2015)
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