Reversible Competitive α-Ketoheterocycle Inhibitors Of Fatty Acid Amide Hydrolase Containing Additional Conformational Constraints In The Acyl Side Chain: Orally Active, Long-Acting Analgesics
Cyrine Ezzili, Mauro Mileni, Nicholas McGlinchey, Jonathan Z. Long, Steven G. Kinsey, Dustin G. Hochstatter, Raymond C. Stevens, Aron H. Lichtman, Benjamin F. Cravatt, Edward J. Bilsky, Dale L. Boger